SCHEMBL28660406

SCHEMBL28660406

Cc1nc(-c2ccnc(N)c2)sc1C(=O)O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.60
KDM4E B2RXH2 4/20 0.58
RAB9A P51151 3/20 0.58
GAA P10253 2/20 0.58
CDC7 O00311 2/20 0.58
DBF4 Q9UBU7 2/20 0.58
NPC1 O15118 1/20 0.56
POLB P06746 1/20 0.56
ALDH1A1 P00352 3/20 0.54
KMT2A Q03164 2/20 0.53
TARBP2 Q15633 2/20 0.50
GSK3B P49841 1/20 0.50
XDH P47989 4/20 0.47
ABCC4 O15439 1/20 0.47
ABCB11 O95342 1/20 0.47
PGR P06401 1/20 0.47
CHRM1 P11229 1/20 0.47
PDE4A P27815 1/20 0.47
BLVRB P30043 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28658387 0.85 SMN1; SMN2 (0.58) SMN1; SMN2KDM4ERAB9AGAACDC7
SCHEMBL28654454 0.83 CDC7 (0.57) SMN1; SMN2KDM4ERAB9AGAACDC7
SCHEMBL27875453 0.81 CDC7 (0.63) SMN1; SMN2KDM4ERAB9AGAACDC7
SCHEMBL28660397 0.80 SMN1; SMN2 (0.56) SMN1; SMN2KDM4ERAB9AGAANPC1
SCHEMBL3328924 0.79 SMN1; SMN2 (0.76) SMN1; SMN2KDM4ERAB9AGAACDC7
SCHEMBL12582103 0.79 SMN1; SMN2 (0.70) SMN1; SMN2KDM4ERAB9AGAANPC1
SCHEMBL28656962 0.79 KDM4E (0.52) SMN1; SMN2KDM4ERAB9AGAACDC7
SCHEMBL14018508 0.78 RAB9A (0.77) SMN1; SMN2KDM4ERAB9AGAANPC1
SCHEMBL21156699 0.77 RAB9A (0.69) SMN1; SMN2KDM4ERAB9AGAANPC1
SCHEMBL623016 0.76 CDC7 (0.51) SMN1; SMN2RAB9AGAACDC7DBF4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113024534-A 2-pyridylthiazole derivatives and use thereof 武汉光谷亚太医药研究院有限公司 2021-06-25 CN claimed
CN-113024534-B 2-pyridylthiazole derivatives and use thereof 武汉光谷亚太医药研究院有限公司 2023-03-21 CN disclosed
CN-113024534-A 2-pyridylthiazole derivatives and use thereof 武汉光谷亚太医药研究院有限公司 2021-06-25 CN disclosed