SCHEMBL28665677

SCHEMBL28665677

NC(=O)c1cccc(-c2ccccc2)c1-c1nnn[nH]1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.51
KEAP1 Q14145 1/20 0.43
NFE2L2 Q16236 1/20 0.43
PARP1 P09874 7/20 0.43
HNF4A P41235 1/20 0.42
DHODH Q02127 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
CSNK1A1 P48729 2/20 0.40
DYRK1B Q9Y463 2/20 0.40
TYRO3 Q06418 1/20 0.40
IKBKB O14920 1/20 0.39
CHUK O15111 1/20 0.39
IKBKE Q14164 1/20 0.39
PKMYT1 Q99640 1/20 0.39
AURKA O14965 1/20 0.38
PDK2 Q15119 1/20 0.37
CASP1 P29466 1/20 0.37
CCNE2 O96020 1/20 0.37
CDK4 P11802 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4532599 0.89 HNF4A (0.51) BCAT2HNF4ADHODHNPC1RAB9A
SCHEMBL4950797 0.85 BCAT2 (0.36) BCAT2KEAP1NFE2L2PARP1DHODH
SCHEMBL3914195 0.84 BCAT2 (0.41) BCAT2KEAP1NFE2L2PARP1DHODH
SCHEMBL3914170 0.83 CSNK1A1 (0.44) BCAT2KEAP1NFE2L2PARP1DHODH
SCHEMBL6775090 0.82 CYP1A2 (0.43) IKBKBCCNE2CDK4CCND1CCNE1
SCHEMBL2650295 0.81 CSNK1A1 (0.54) BCAT2KEAP1NFE2L2PARP1NPC1
SCHEMBL4950617 0.81 BCAT2 (0.54) BCAT2PARP1DHODHNPC1RAB9A
SCHEMBL6782270 0.80 CCNE2 (0.41) PARP1DHODHCCNE2CDK4CCND1
SCHEMBL11968815 0.79 POLB (0.42) HNF4ADHODHNPC1RAB9AKDR
SCHEMBL27761645 0.79 FGFR1 (0.41) NPC1RAB9ACSNK1A1DYRK1BMAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107922394-B 3-tetrazolyl-benzene-1, 2-disulfonamide derivatives as metallo-beta-lactamase inhibitors 默沙东公司 2021-07-13 CN disclosed