SCHEMBL28668261

SCHEMBL28668261

CN(c1ccc2c(cnn2C(=O)O)c1)c1ccnc(Cl)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 2/20 0.41
CHEK1 O14757 1/20 0.37
AURKA O14965 1/20 0.37
DAPK3 O43293 1/20 0.37
CSNK1A1 P48729 1/20 0.37
GSK3A P49840 1/20 0.37
LIMK1 P53667 1/20 0.37
IKBKE Q14164 1/20 0.37
MAPK14 Q16539 1/20 0.37
TAOK1 Q7L7X3 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
DYRK1B Q9Y463 1/20 0.37
MAPT P10636 2/20 0.36
KMT2A Q03164 3/20 0.35
RAB9A P51151 3/20 0.34
SHMT2 P34897 2/20 0.34
RXRA P19793 4/20 0.34
RXRB P28702 3/20 0.34
HDAC3 O15379 2/20 0.33
HDAC1 Q13547 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15638766 0.85 ROCK2 (0.42) SLC22A12CHEK1AURKADAPK3CSNK1A1
SCHEMBL28336523 0.81 SLC22A12 (0.36) SLC22A12CHEK1AURKADAPK3CSNK1A1
SCHEMBL10187295 0.78 KDR (0.42) AURKALIMK1TAOK1RXRARXRB
SCHEMBL15514657 0.73 RXRA (0.41) AURKAMAPTRAB9ARXRARXRB
SCHEMBL15639911 0.73 ROCK2 (0.42) SLC22A12CHEK1AURKADAPK3CSNK1A1
SCHEMBL5227351 0.73 KDR (0.44) AURKACSNK1A1TAOK1CLK4RAB9A
SCHEMBL12185524 0.72 KDR (0.39) MAPTKMT2ARAB9ANPC1MEN1
SCHEMBL15514096 0.72 RXRA (0.39) AURKARXRARXRBHDAC3HDAC1
SCHEMBL17025789 0.72 CDC7 (0.48) SLC22A12CHEK1AURKADAPK3CSNK1A1
SCHEMBL27925382 0.71 RXRA (0.38) AURKARXRARXRBRXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113773308-A RHO kinase inhibitors 卡德门企业有限公司 2021-12-10 CN disclosed
CN-113637008-A RHO kinase inhibitors 卡德门企业有限公司 2021-11-12 CN disclosed
CN-113637007-A RHO kinase inhibitors 卡德门企业有限公司 2021-11-12 CN disclosed
CN-113620933-A RHO kinase inhibitors 卡德门企业有限公司 2021-11-09 CN disclosed