SCHEMBL28668564

SCHEMBL28668564

CC(NC(=O)OC(C)(C)C)C(=O)N1Cc2ccccc2C1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 8/20 0.51
CTSK P43235 1/20 0.47
DPP8 Q6V1X1 3/20 0.47
DPP9 Q86TI2 3/20 0.47
DPP7 Q9UHL4 2/20 0.47
ATM Q13315 2/20 0.47
DPP4 P27487 1/20 0.47
KCNH2 Q12809 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
MAPK1 P28482 1/20 0.45
NOTUM Q6P988 1/20 0.45
HRH2 P25021 1/20 0.44
HRH1 P35367 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29758946 1.00 NAMPT (0.51) NAMPTCTSKDPP8DPP9DPP7
SCHEMBL18212438 1.00 NAMPT (0.51) NAMPTCTSKDPP8DPP9DPP7
SCHEMBL28650975 0.91 CTSK (0.56) CTSKATMHRH3NOTUM
SCHEMBL29758964 0.91 CTSK (0.56) CTSKATMHRH3NOTUM
SCHEMBL18215088 0.91 CTSK (0.56) CTSKATMHRH3NOTUM
SCHEMBL6164761 0.82 KMT2A (0.60) CTSKDPP8DPP9ATMMAPK1
SCHEMBL8244870 0.82 KMT2A (0.60) CTSKDPP8DPP9ATMMAPK1
SCHEMBL10739004 0.81 ACE (0.59)
SCHEMBL27705686 0.81 ACE (0.59)
SCHEMBL31039670 0.80 DRD2 (0.43) NAMPTCTSKDPP8DPP9DPP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107735088-B Histone deacetylase inhibitors, compositions and methods of use thereof CHDI基金会股份有限公司 2021-11-02 CN disclosed