SCHEMBL28670141

SCHEMBL28670141

COC(=O)c1c(O)cc(OC)cc1/C=C/c1ccc(O)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 1/20 0.56
DPP4 P27487 1/20 0.56
NFKB2 Q00653 1/20 0.56
RELA Q04206 1/20 0.56
CYP1A1 P04798 3/20 0.56
CYP1B1 Q16678 3/20 0.56
TTR P02766 2/20 0.56
ALOX5 P09917 2/20 0.56
PTGS2 P35354 2/20 0.56
MAPT P10636 2/20 0.56
KDM4E B2RXH2 1/20 0.56
MEN1 O00255 1/20 0.56
NPC1 O15118 1/20 0.56
ABL1 P00519 1/20 0.56
ABCB1 P08183 1/20 0.56
GAA P10253 1/20 0.56
BCR P11274 1/20 0.56
NQO2 P16083 1/20 0.56
PTGS1 P23219 1/20 0.56
MAPK1 P28482 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28670143 1.00 NFKB1 (0.56) NFKB1DPP4NFKB2RELACYP1A1
SCHEMBL16191726 0.94 SLC5A1 (0.57) NFKB1DPP4NFKB2RELACYP1A1
SCHEMBL16191723 0.94 SLC5A1 (0.57) NFKB1DPP4NFKB2RELACYP1A1
SCHEMBL16191523 0.92 CYP3A4 (0.55) NFKB1DPP4NFKB2RELACYP1A1
SCHEMBL16191525 0.92 CYP3A4 (0.55) NFKB1DPP4NFKB2RELACYP1A1
SCHEMBL16191660 0.91 NQO2 (0.52) NFKB1DPP4NFKB2RELACYP1A1
SCHEMBL16191657 0.91 NQO2 (0.52) NFKB1DPP4NFKB2RELACYP1A1
SCHEMBL16191921 0.90 MAOA (0.63) NFKB1DPP4NFKB2RELACYP1A1
SCHEMBL16191751 0.90 MAOA (0.63) NFKB1DPP4NFKB2RELACYP1A1
SCHEMBL30358574 0.89 ALOX5 (0.58) RELATTRALOX5PTGS2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116270577-A Application of polysubstituted benzene compounds in preparation of medicines for treating cognitive impairment diseases, structure and preparation method 中国医学科学院医药生物技术研究所 2023-06-23 CN disclosed
CN-116270576-A Application of polysubstituted benzene compounds in preparation of medicines for treating cognitive impairment diseases, structure and preparation method 中国医学科学院医药生物技术研究所 2023-06-23 CN disclosed
CN-113521048-B Application of polysubstituted benzene compound in preparation of medicine for treating cognitive disorder diseases, structure and preparation method 中国医学科学院医药生物技术研究所 2023-04-14 CN disclosed
CN-113521048-A Application of polysubstituted benzene compound in preparation of medicine for treating cognitive disorder diseases, structure and preparation method 中国医学科学院医药生物技术研究所 2021-10-22 CN disclosed