SCHEMBL286702

SCHEMBL286702

COC(=O)Cc1cccc(Br)c1OC

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.48
MEN1 O00255 2/20 0.48
KDM4E B2RXH2 5/20 0.43
ALDH1A1 P00352 4/20 0.40
TDP1 Q9NUW8 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
HTR2A P28223 1/20 0.39
TSHR P16473 1/20 0.39
PPARG P37231 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
MAPT P10636 2/20 0.38
GAA P10253 1/20 0.38
CYP4F2 P78329 1/20 0.38
CYP4A11 Q02928 1/20 0.38
HSD17B10 Q99714 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2729290 0.85 MEN1 (0.49) KMT2AMEN1KDM4EALDH1A1TDP1
SCHEMBL31111007 0.84 PTPN1 (0.40) KMT2AMEN1KDM4EALDH1A1TDP1
SCHEMBL27287731 0.84 MTNR1A (0.52) KMT2AMEN1KDM4EALDH1A1TDP1
SCHEMBL14420215 0.83 KDM4E (0.44) KMT2AMEN1KDM4EALDH1A1TDP1
SCHEMBL31042998 0.82 KMT2A (0.51) KMT2AMEN1KDM4EALDH1A1TDP1
SCHEMBL965852 0.82 KMT2A (0.51) KMT2AMEN1KDM4EALDH1A1TDP1
SCHEMBL23703592 0.82 KDM4E (0.43) KMT2AMEN1KDM4EALDH1A1TDP1
SCHEMBL2060569 0.81 KDM4E (0.44) KMT2AMEN1KDM4EALDH1A1TDP1
SCHEMBL13696433 0.81 SMN1; SMN2 (0.46) KMT2AKDM4EALDH1A1TDP1L3MBTL1
SCHEMBL15056307 0.81 KDM4E (0.44) KMT2AMEN1KDM4EALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4298135-B1 BIS-PHENOXY-ETHER LIGANDS FOR GROUP IV POLYOLEFIN CATALYSIS DOW GLOBAL TECHNOLOGIES LLC (US) 2025-04-16 EP disclosed
US-20240158542-A1 BIS-PHENOXY-ETHER LIGANDS FOR GROUP IV POLYOLEFIN CATALYSIS DOW GLOBAL TECHNOLOGIES LLC (US) 2024-05-16 US disclosed
CN-117580836-A Pyrimidine ring structure derivative and application thereof 四川汇宇制药股份有限公司 2024-02-20 CN disclosed
EP-4298135-A1 BIS-PHENOXY-ETHER LIGANDS FOR GROUP IV POLYOLEFIN CATALYSIS Dow Global Technologies LLC (US) 2024-01-03 EP disclosed
CN-116897168-A Bis-phenoxy-ether ligands for Group IV polyolefin catalysis 陶氏环球技术有限责任公司 2023-10-17 CN disclosed
WO-2022268209-A1 DERIVATIVE HAVING PYRIMIDINE-FUSED CYCLIC STRUCTURE, AND USE THEREOF 四川汇宇制药股份有限公司 2022-12-29 WO disclosed
WO-2022268209-A1 DERIVATIVE HAVING PYRIMIDINE-FUSED CYCLIC STRUCTURE, AND USE THEREOF 四川汇宇制药股份有限公司 2022-12-29 WO disclosed
WO-2022183005-A1 BIS-PHENOXY-ETHER LIGANDS FOR GROUP IV POLYOLEFIN CATALYSIS DOW GLOBAL TECHNOLOGIES LLC (US) 2022-09-01 WO disclosed
CN-105143170-B For treating the aromatic compounds of pulmonary fibrosis, liver fibrosis, fibrosis of skin and cardiac fibrosis being substituted 普罗米蒂克医药SMT有限公司 2019-11-08 CN disclosed
EP-2794563-B1 HETEROCYCLYL DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2017-02-22 EP disclosed
US-9255090-B2 Heterocyclyl derivatives and their use as prostaglandin D2 receptor modulators ACTELION PHARMACEUTICALS LTD. (CH) 2016-02-09 US disclosed
US-20150252036-A1 Heterocyclyl Derivatives and their use as Prostaglandin D2 Receptor Modulators IDORSIA PHARMACEUTICALS LTD (CH) 2015-09-10 US disclosed
EP-2794563-A1 HETEROCYCLYL DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS Actelion Pharmaceuticals Ltd. (CH) 2014-10-29 EP disclosed
WO-2013093842-A1 HETEROCYCLYL DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2013-06-27 WO disclosed
EP-2427444-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL Merck Sharp & Dohme Corp. (US) 2012-03-14 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150252036-A1 Heterocyclyl Derivatives and their use as Prostaglandin D2 Receptor Modulators PTGDR, PTGER1, PTGDR2 KMT2A 4057/4885MEN1 2511/4885KDM4E 4188/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.