SCHEMBL28670748

SCHEMBL28670748

CC(C)(C)[Si](C)(C)O[C@@H]1C[C@H](c2cccc(F)c2)N(c2cccnc2)C1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 2/20 0.37
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CHRNB2 P17787 4/20 0.34
CHRNA4 P43681 4/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
JAK2 O60674 1/20 0.34
NTRK1 P04629 1/20 0.34
PDE5A O76074 1/20 0.34
DPP4 P27487 1/20 0.34
NR3C2 P08235 1/20 0.34
PIK3CD O00329 1/20 0.34
PIK3R1 P27986 1/20 0.34
SLC6A9 P48067 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL455586 0.79 RIPK1 (0.40) RIPK1MAOAMAOBJAK2NTRK1
SCHEMBL981085 0.74 RIPK1 (0.34) RIPK1MAOAMAOBJAK2NTRK1
SCHEMBL448624 0.73 RIPK1 (0.47) RIPK1MAOAMAOBJAK2NTRK1
SCHEMBL430776 0.73 RIPK1 (0.47) RIPK1MAOAMAOBJAK2NTRK1
SCHEMBL945868 0.69 NTRK1 (0.58) JAK2NTRK1
SCHEMBL4518142 0.67 RIPK1 (0.41) RIPK1MAOAMAOBPDE5A
SCHEMBL4501581 0.67 RIPK1 (0.41) RIPK1MAOAMAOBPDE5A
SCHEMBL433152 0.67 HTR2A (0.35) RIPK1MAOAMAOB
SCHEMBL431587 0.67 HTR2A (0.35) RIPK1MAOAMAOB
SCHEMBL451170 0.67 HTR2A (0.35) RIPK1MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110003214-B Substituted pyrazolo [1,5-a ] pyrimidine compounds as TRK kinase inhibitors 阵列生物制药公司 2021-12-21 CN disclosed