SCHEMBL28670769

SCHEMBL28670769

O=[N+]([O-])c1ccc(Oc2ccc(C34CC5CC(CC(C5)C3)C4)cc2Cl)cc1

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE7A Q13946 1/20 0.53
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
ALDH1A1 P00352 6/20 0.47
MAPT P10636 3/20 0.47
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
GAA P10253 1/20 0.46
PKM P14618 1/20 0.46
PGR P06401 1/20 0.46
HSPB1 P04792 2/20 0.43
KDM4E B2RXH2 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.41
FAAH O00519 1/20 0.39
GPR55 Q9Y2T6 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31168053 1.00 PDE7A (0.53) PDE7ANPC1RAB9AALDH1A1MAPT
SCHEMBL22452613 0.85 PDE7A (0.48) PDE7ANPC1RAB9AALDH1A1MAPT
SCHEMBL15071010 0.83 RAB9A (0.59) NPC1RAB9AALDH1A1MAPTMEN1
SCHEMBL22453327 0.81 ALDH1A1 (0.55) PDE7ARAB9AALDH1A1MAPTMEN1
SCHEMBL15071008 0.81 HSPB1 (0.55) PDE7ANPC1RAB9AALDH1A1MAPT
SCHEMBL16049433 0.79 HSPB1 (0.46) PDE7ANPC1RAB9AALDH1A1MAPT
SCHEMBL3190249 0.79 NPC1 (0.45) PDE7ANPC1RAB9AALDH1A1MAPT
SCHEMBL18992722 0.77 NPC1 (0.69) NPC1RAB9AALDH1A1MAPTMEN1
SCHEMBL28015555 0.77 ALDH1A1 (0.44) PDE7ANPC1RAB9AALDH1A1MAPT
SCHEMBL30354727 0.76 NPC1 (0.49) NPC1RAB9AALDH1A1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113811300-A Novel small molecule inhibitors of TEAD transcription factor 总医院公司 2021-12-17 CN disclosed