SCHEMBL286709

SCHEMBL286709

CCCCc1noc(C)c1COc1cc(C(=O)OC(C)C(N)=O)n(C)n1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.40
ALDH1A1 P00352 4/20 0.34
HTT P42858 2/20 0.34
GABRA5 P31644 3/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
USP2 O75604 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
MEN1 O00255 1/20 0.33
GABRA1 P14867 2/20 0.33
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
TAS2R8 Q9NYW2 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL286377 0.88 GABRA5 (0.39) KMT2AALDH1A1HTTGABRA5L3MBTL1
SCHEMBL286143 0.86 ALDH1A1 (0.35) KMT2AALDH1A1GABRA5L3MBTL1SMN1; SMN2
SCHEMBL286369 0.85 NR1H4 (0.40) HTTGABRA5L3MBTL1GAAGABRA1
SCHEMBL285772 0.84 GABRA5 (0.42) GABRA5GABRA1
SCHEMBL286209 0.81 GABRA5 (0.44) GABRA5GABRA1
SCHEMBL286328 0.81 KMT2A (0.38) KMT2AALDH1A1HTTGABRA5L3MBTL1
SCHEMBL286582 0.81 KMT2A (0.38) KMT2AALDH1A1HTTGABRA5L3MBTL1
SCHEMBL285773 0.80 POLB (0.40) GABRA5L3MBTL1GABRA1TAS2R8
SCHEMBL286425 0.80 GABRA5 (0.52) GABRA5GABRA1
SCHEMBL286045 0.80 GABRA5 (0.52) GABRA5GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427455-A1 ISOXAZOLE-PYRAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2012-03-14 EP disclosed