SCHEMBL28673167

SCHEMBL28673167

COC(=O)c1cc(C)cn1Cc1ccncc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.55
MAPK10 P53779 1/20 0.55
GAA P10253 3/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
NPSR1 Q6W5P4 1/20 0.45
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44
CCNC P24863 1/20 0.43
CDK8 P49336 1/20 0.43
CYP46A1 Q9Y6A2 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
MAPT P10636 2/20 0.41
TSHR P16473 1/20 0.41
LMNA P02545 1/20 0.41
DNM1L O00429 1/20 0.41
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24937330 0.85 MAPK10 (0.54) USP2MAPK10GAAL3MBTL1NPSR1
SCHEMBL24435291 0.83 MAPK10 (0.52) USP2MAPK10GAAL3MBTL1NPSR1
SCHEMBL16116241 0.79 CCNC (0.71) USP2MAPK10NPSR1CYP11B1CYP11B2
SCHEMBL25395065 0.77 USP2 (0.51) USP2MAPK10CYP11B1CYP11B2HDAC3
SCHEMBL28683880 0.77 CYP11B1 (0.70) USP2MAPK10CYP11B1CYP11B2TSHR
SCHEMBL24434966 0.75 RAB9A (0.58) USP2MAPK10GAAL3MBTL1NPSR1
SCHEMBL28689329 0.74 MEN1 (0.49) USP2MAPK10GAAL3MBTL1NPSR1
SCHEMBL1562627 0.73 SMN1; SMN2 (0.54) GAAMAPTTSHRLMNAKDM4E
SCHEMBL28932115 0.73 MAPK10 (0.50) USP2MAPK10GAACYP11B1CYP11B2
SCHEMBL11914100 0.73 ABL1 (0.48) GAAL3MBTL1NPSR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3930849-B1 THIAZOLE DERIVATIVES AS PROTEIN SECRETION INHIBITORS KEZAR LIFE SCIENCES (US) 2025-02-19 EP disclosed
CN-113993587-A Thiazole derivatives as protein secretion inhibitors 科智生命科学公司 2022-01-28 CN disclosed