SCHEMBL28679752

SCHEMBL28679752

C=C1C=CC(C(=O)OCC)=CN(C(=O)OC(C)(C)C)C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.40
GLA P06280 1/20 0.39
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
ALDH1A1 P00352 3/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
TP53 P04637 1/20 0.33
POLB P06746 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
GPR119 Q8TDV5 1/20 0.33
ATM Q13315 1/20 0.32
CRHBP P24387 1/20 0.32
CRHR2 Q13324 1/20 0.32
AKR1C3 P42330 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28670678 0.73 GLA (0.39) ADORA1GLAMEN1KMT2AALDH1A1
SCHEMBL4777248 0.72 GLA (0.36) ADORA1GLAMEN1KMT2AALDH1A1
SCHEMBL27037069 0.71 ESR2 (0.36) ADORA1MEN1KMT2ASMN1; SMN2GPR119
SCHEMBL20670426 0.70 GLA (0.42) ADORA1GLAMEN1KMT2AALDH1A1
SCHEMBL29099338 0.69 GLA (0.43) ADORA1GLAMEN1KMT2AALDH1A1
SCHEMBL7863282 0.69 GLA (0.46) ADORA1GLAMEN1KMT2AALDH1A1
SCHEMBL28970107 0.68 PREP (0.36) MEN1KMT2AALDH1A1LMNASMN1; SMN2
SCHEMBL3505154 0.67 ESR2 (0.45) ADORA1MEN1KMT2ASMN1; SMN2GPR119
SCHEMBL28679745 0.66 ADORA1 (0.40) ADORA1GLAMEN1KMT2AALDH1A1
SCHEMBL28932778 0.66 ADORA1 (0.38) ADORA1GLAMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113795491-A Bridged ring-3, 4-dihydro-pyrido [1,2-a ] pyrazine-1, 8-dione compound and pharmaceutical use thereof 上海拓界生物医药科技有限公司 2021-12-14 CN disclosed