SCHEMBL28680289

SCHEMBL28680289

CCOC(=O)C1=C(O)C(=O)N(c2cccc3cccc(Cl)c23)CCC1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
CASP3 P42574 4/20 0.40
KDM4E B2RXH2 2/20 0.39
MAPK1 P28482 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
PDE4B Q07343 1/20 0.38
ALOX5 P09917 1/20 0.38
CHRM2 P08172 1/20 0.37
CHRM4 P08173 1/20 0.37
CHRM5 P08912 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30887665 1.00 ALDH1A1 (0.43) ALDH1A1MEN1KMT2ACASP3KDM4E
SCHEMBL28680301 0.84 CASP3 (0.56) ALDH1A1MEN1KMT2ACASP3KDM4E
SCHEMBL28688250 0.67 MAPT (0.36) ALDH1A1MEN1KMT2AKDM4EMAPK1
SCHEMBL30887637 0.67 MAPT (0.36) ALDH1A1MEN1KMT2AKDM4EMAPK1
SCHEMBL12202083 0.66 CASP3 (0.45) ALDH1A1MEN1KMT2ACASP3KDM4E
SCHEMBL8654624 0.65 GAA (0.45) ALDH1A1MEN1KMT2AKDM4EMAPK1
SCHEMBL9208732 0.64 CASP3 (0.66) ALDH1A1CASP3KDM4ECHRM2CHRM4
SCHEMBL30671499 0.64 KDM4E (0.37) ALDH1A1MEN1KMT2AKDM4ECHRM2
SCHEMBL1280809 0.63 HSD17B10 (0.54) ALDH1A1MEN1KMT2AKDM4EMAPK1
SCHEMBL24970169 0.62 ALDH1A1 (0.42) ALDH1A1MEN1KMT2AKDM4EMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113135924-B Pyrimidine derivatives and their use in medicine 广东东阳光药业股份有限公司 2024-04-26 CN disclosed
CN-113135924-A Pyrimidine derivatives and their use in medicine 广东东阳光药业有限公司 2021-07-20 CN disclosed