SCHEMBL28680301

SCHEMBL28680301

CCOC(=O)C1=C(O)C(=O)N(c2cccc3ccccc23)CCC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.56
KMT2A Q03164 5/20 0.43
MEN1 O00255 3/20 0.43
ALDH1A1 P00352 3/20 0.43
CDC25B P30305 3/20 0.42
KDM4E B2RXH2 3/20 0.42
MAPT P10636 1/20 0.42
HTT P42858 1/20 0.42
RECQL P46063 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
PKM P14618 1/20 0.41
ALOX5 P09917 1/20 0.40
CDC25A P30304 1/20 0.40
CDC25C P30307 1/20 0.40
POLB P06746 1/20 0.39
CHRM2 P08172 1/20 0.39
CHRM4 P08173 1/20 0.39
CHRM5 P08912 1/20 0.39
CHRM1 P11229 1/20 0.39
CHRM3 P20309 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30887665 0.84 ALDH1A1 (0.43) CASP3KMT2AMEN1ALDH1A1KDM4E
SCHEMBL28680289 0.84 ALDH1A1 (0.43) CASP3KMT2AMEN1ALDH1A1KDM4E
SCHEMBL3265630 0.72 MAPT (0.64) CASP3KMT2AMEN1ALDH1A1CDC25B
SCHEMBL27792820 0.72 CASP3 (1.00) CASP3ALOX15
SCHEMBL12202083 0.71 CASP3 (0.45) CASP3KMT2AMEN1ALDH1A1KDM4E
SCHEMBL8654624 0.70 GAA (0.45) KMT2AMEN1ALDH1A1KDM4EMAPT
SCHEMBL9208732 0.69 CASP3 (0.66) CASP3ALDH1A1KDM4EMAPTCHRM2
SCHEMBL611001 0.68 SCN9A (0.47) ALDH1A1KDM4EMAPTPKMPOLB
SCHEMBL29741442 0.68 SCN9A (0.47) ALDH1A1KDM4EMAPTPKMPOLB
SCHEMBL29929651 0.68 SCN9A (0.47) ALDH1A1KDM4EMAPTPKMPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113135924-B Pyrimidine derivatives and their use in medicine 广东东阳光药业股份有限公司 2024-04-26 CN disclosed
CN-113135924-A Pyrimidine derivatives and their use in medicine 广东东阳光药业有限公司 2021-07-20 CN disclosed