SCHEMBL28680774

SCHEMBL28680774

O=C(COCc1cccc(F)c1)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 2/20 0.56
MAOB P27338 3/20 0.51
HCAR2 Q8TDS4 1/20 0.50
PARP10 Q53GL7 1/20 0.49
PPARA Q07869 1/20 0.48
IDO1 P14902 2/20 0.47
AGXT P21549 2/20 0.47
KDM4E B2RXH2 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
MAPT P10636 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
MRGPRX4 Q96LA9 3/20 0.46
LMNA P02545 1/20 0.46
MAPK1 P28482 1/20 0.46
CASP3 P42574 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
SENP6 Q9GZR1 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28680772 0.91 NR4A2 (0.49) NR4A2MAOBHCAR2KDM4EMAPT
SCHEMBL7809052 0.85 NR4A2 (0.53) NR4A2MAOBHCAR2PARP10PPARA
SCHEMBL360528 0.84 NR4A2 (0.55) NR4A2MAOBHCAR2PARP10PPARA
SCHEMBL657234 0.84 TDP1 (0.55) KDM4ECYP1A2MAPTCYP2C9MAPK1
SCHEMBL27622766 0.83 LMNA (0.60) NR4A2MAOBKDM4EMAPTLMNA
SCHEMBL4888735 0.82 NR4A2 (0.56) NR4A2MAOBHCAR2IDO1AGXT
SCHEMBL8888362 0.79 MRGPRX4 (0.57) MAOBIDO1AGXTCYP1A2MRGPRX4
SCHEMBL11439089 0.79 LOXL2 (0.57) KDM4EMAPTMRGPRX4LMNARAB9A
SCHEMBL570730 0.79 MAPT (0.51) NR4A2MAPTL3MBTL1GPR52RAB9A
SCHEMBL7646959 0.78 MEN1 (0.54) NR4A2HCAR2PPARAKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109020883-B 3-cyano-2-aminopyridine derivative and preparation method and application thereof 广西民族大学 2022-02-08 CN disclosed