SCHEMBL28684201

SCHEMBL28684201

COC(=O)CCCCCCNC(=O)c1ccc(C(=O)CBr)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.56
RAB9A P51151 2/20 0.56
MAPK1 P28482 1/20 0.55
ALDH1A1 P00352 1/20 0.53
POLB P06746 2/20 0.50
THRA P10827 1/20 0.50
THRB P10828 1/20 0.50
LMNA P02545 2/20 0.48
MAPT P10636 1/20 0.48
HTT P42858 1/20 0.48
HDAC3 O15379 6/20 0.48
HDAC1 Q13547 6/20 0.48
HDAC2 Q92769 6/20 0.48
HDAC6 Q9UBN7 6/20 0.48
HDAC4 P56524 5/20 0.48
HDAC7 Q8WUI4 5/20 0.48
HDAC10 Q969S8 5/20 0.48
HDAC11 Q96DB2 5/20 0.48
HDAC8 Q9BY41 5/20 0.48
HDAC9 Q9UKV0 5/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28693969 1.00 NPC1 (0.56) NPC1RAB9AMAPK1ALDH1A1POLB
SCHEMBL28693966 0.99 ALDH1A1 (0.54) NPC1RAB9AMAPK1ALDH1A1POLB
SCHEMBL450259 0.86 NPC1 (0.59) NPC1RAB9AMAPK1ALDH1A1POLB
SCHEMBL2631174 0.84 L3MBTL1 (0.68) NPC1RAB9AMAPK1ALDH1A1POLB
SCHEMBL28706039 0.84 NPC1 (0.60) NPC1RAB9AMAPK1ALDH1A1POLB
SCHEMBL28706800 0.84 NPC1 (0.60) NPC1RAB9AMAPK1ALDH1A1POLB
SCHEMBL1233065 0.83 NPC1 (0.82) NPC1RAB9AMAPK1ALDH1A1POLB
SCHEMBL4954251 0.83 NPC1 (0.59) NPC1RAB9AMAPK1ALDH1A1POLB
SCHEMBL1232846 0.83 NPC1 (0.59) NPC1RAB9AMAPK1ALDH1A1POLB
SCHEMBL12672001 0.82 NAAA (0.67) NPC1RAB9AMAPK1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114075187-B Carbonyl pyrazole antitumor compound as well as preparation method and application thereof 山东大学 2023-05-12 CN disclosed
CN-114075187-A Carbonyl pyrazole anti-tumor compound and preparation method and application thereof 山东大学 2022-02-22 CN disclosed