SCHEMBL28684283

SCHEMBL28684283

O=c1[nH]c2ccc([N+](=O)[O-])cc2c(=O)n1Cc1ccccc1

nearest known ligand 0.80

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.62
ALDH1A1 P00352 2/20 0.62
HPGD P15428 1/20 0.62
SMN1; SMN2 Q16637 1/20 0.62
PGR P06401 1/20 0.61
CA12 O43570 1/20 0.60
CA9 Q16790 1/20 0.60
MEN1 O00255 3/20 0.58
KMT2A Q03164 3/20 0.58
CTSV O60911 3/20 0.53
CTSL P07711 3/20 0.53
PARP1 P09874 1/20 0.52
DHFR P00374 1/20 0.52
KAT2B Q92831 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28932143 0.87 CA12 (0.51) KDM4EALDH1A1HPGDSMN1; SMN2PGR
SCHEMBL7650431 0.86 KDM4E (0.65) KDM4ECA12CA9MEN1KMT2A
SCHEMBL10745767 0.83 CA12 (0.61) ALDH1A1SMN1; SMN2PGRCA12CA9
SCHEMBL17434518 0.83 CA12 (0.64) ALDH1A1CA12CA9MEN1KMT2A
SCHEMBL28694312 0.82 KDM4E (0.56) KDM4EALDH1A1HPGDSMN1; SMN2CA12
SCHEMBL29428154 0.82 KDM4E (0.56) KDM4EALDH1A1HPGDSMN1; SMN2CA12
SCHEMBL28683072 0.81 MEN1 (0.58) ALDH1A1HPGDPGRMEN1KMT2A
SCHEMBL28700145 0.79 VCAM1 (0.47) ALDH1A1SMN1; SMN2CA12CA9MEN1
SCHEMBL28932333 0.79 ALDH1A1 (0.68) KDM4EALDH1A1HPGDSMN1; SMN2PGR
SCHEMBL10085009 0.79 KDM4E (0.68) KDM4EALDH1A1HPGDSMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109776434-B 3-benzyl-6-acylamino-2, 4- (1H,3H) -quinazoline diketone derivative and synthesis method and application thereof 中南大学 2022-01-28 CN disclosed