SCHEMBL28685463

SCHEMBL28685463

Clc1ccc2oc(C3CCCN3)nc2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.49
CDC7 O00311 1/20 0.49
CIT O14578 1/20 0.49
PIM1 P11309 1/20 0.49
CSNK2A2 P19784 1/20 0.49
GSK3B P49841 1/20 0.49
CSNK2B P67870 1/20 0.49
CSNK2A1 P68400 1/20 0.49
DYRK1A Q13627 1/20 0.49
CSNK2A3 Q8NEV1 1/20 0.49
TAOK3 Q9H2K8 1/20 0.49
CHRNB2 P17787 1/20 0.46
CHRNA4 P43681 1/20 0.46
PSMB8 P28062 1/20 0.46
LMNA P02545 3/20 0.45
MAPT P10636 2/20 0.45
THRB P10828 1/20 0.45
ALOX15 P16050 1/20 0.45
MAPK1 P28482 1/20 0.45
ALDH1A1 P00352 4/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24359797 0.85 PSMB8 (0.44) CYP1A2CDC7CITPIM1CSNK2A2
SCHEMBL28686943 0.83 MPO (0.60) CYP1A2CDC7CITPIM1CSNK2A2
SCHEMBL28901276 0.80 CHRNB2 (0.54) CYP1A2CHRNB2CHRNA4LMNACYP2C19
SCHEMBL28901281 0.80 CHRNB2 (0.54) CYP1A2CHRNB2CHRNA4LMNACYP2C19
SCHEMBL12649101 0.80 CHRNB2 (0.54) CYP1A2CHRNB2CHRNA4LMNACYP2C19
SCHEMBL14555059 0.78 MPO (0.61) CYP1A2CDC7PIM1CSNK2BCSNK2A1
SCHEMBL29688673 0.77 MPO (0.59) CYP1A2PSMB8LMNAMAPTTHRB
SCHEMBL4712528 0.77 MPO (0.59) CYP1A2PSMB8LMNAMAPTTHRB
SCHEMBL7850149 0.76 CHRNB2 (0.60) CYP1A2CDC7CITPIM1CSNK2A2
SCHEMBL7842435 0.76 CHRNB2 (0.60) CYP1A2CDC7CITPIM1CSNK2A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112876479-B Crystalline forms of octahydropyrrolo [3,4-c ] pyrrole derivatives 广东东阳光药业有限公司 2022-07-26 CN disclosed
CN-112876478-B Crystalline forms of octahydropyrrolo [3,4-c ] pyrrole derivatives 广东东阳光药业有限公司 2022-07-26 CN disclosed
CN-112876480-B Crystalline forms of octahydropyrrolo [3,4-c ] pyrrole derivatives 广东东阳光药业有限公司 2022-07-26 CN disclosed
CN-112876481-B Crystalline forms of octahydropyrrolo [3,4-c ] pyrrole derivatives 广东东阳光药业有限公司 2022-07-26 CN disclosed
CN-112876477-B Crystalline forms of octahydropyrrolo [3,4-c ] pyrrole derivatives 广东东阳光药业有限公司 2022-07-26 CN disclosed
CN-109988169-B Octahydropyrrolo [3,4-c ] pyrrole derivatives and uses thereof 广东东阳光药业有限公司 2022-02-01 CN disclosed
CN-112876480-A Crystalline forms of octahydropyrrolo [3,4-c ] pyrrole derivatives 广东东阳光药业有限公司 2021-06-01 CN disclosed
CN-112876478-A Crystalline forms of octahydropyrrolo [3,4-c ] pyrrole derivatives 广东东阳光药业有限公司 2021-06-01 CN disclosed
CN-112876481-A Crystalline forms of octahydropyrrolo [3,4-c ] pyrrole derivatives 广东东阳光药业有限公司 2021-06-01 CN disclosed
CN-112876475-A Salts of octahydropyrrolo [3,4-c ] pyrrole derivatives 广东东阳光药业有限公司 2021-06-01 CN disclosed
CN-112876477-A Crystalline forms of octahydropyrrolo [3,4-c ] pyrrole derivatives 广东东阳光药业有限公司 2021-06-01 CN disclosed
CN-112876479-A Crystalline forms of octahydropyrrolo [3,4-c ] pyrrole derivatives 广东东阳光药业有限公司 2021-06-01 CN disclosed