SCHEMBL28685992

SCHEMBL28685992

COc1ccccc1NC(=O)[C@H]1CCN(C(=O)OC(C)(C)C)C1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.65
BACE1 P56817 1/20 0.65
SMN1; SMN2 Q16637 2/20 0.62
KMT2A Q03164 2/20 0.62
MGLL Q99685 1/20 0.59
KDM4E B2RXH2 2/20 0.58
GAA P10253 1/20 0.56
MAPT P10636 1/20 0.56
TSHR P16473 1/20 0.55
PTPN2 P17706 1/20 0.55
PTPN1 P18031 1/20 0.55
PTPN6 P29350 1/20 0.55
TRPV1 Q8NER1 1/20 0.54
ALDH1A1 P00352 2/20 0.53
LMNA P02545 1/20 0.52
TGFBR1 P36897 1/20 0.52
HSD17B10 Q99714 1/20 0.51
ABL1 P00519 1/20 0.51
RIN1 Q13671 1/20 0.51
STS P08842 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28685994 1.00 ACHE (0.65) ACHEBACE1SMN1; SMN2KMT2AMGLL
SCHEMBL12847604 0.86 PTPN2 (0.57) ACHEBACE1KMT2AKDM4EPTPN2
SCHEMBL26025076 0.83 PTPN2 (0.54) KMT2AKDM4ETSHRPTPN2PTPN1
SCHEMBL30496051 0.83 PTPN2 (0.54) KMT2AKDM4ETSHRPTPN2PTPN1
SCHEMBL25362245 0.83 PTPN2 (0.54) KMT2AKDM4ETSHRPTPN2PTPN1
SCHEMBL742791 0.83 GAA (0.55) ACHEBACE1SMN1; SMN2KMT2AMGLL
SCHEMBL762544 0.83 GAA (0.55) ACHEBACE1SMN1; SMN2KMT2AMGLL
SCHEMBL29686111 0.82 PTPN2 (0.71) ACHEBACE1KDM4EMAPTPTPN2
SCHEMBL1317618 0.82 PTPN2 (0.71) ACHEBACE1KDM4EMAPTPTPN2
SCHEMBL29971632 0.82 PTPN2 (0.71) ACHEBACE1KDM4EMAPTPTPN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113354635-B Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2023-04-18 CN disclosed
CN-113354635-A Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2021-09-07 CN disclosed