SCHEMBL2869174

SCHEMBL2869174

COc1ccc(C(=O)c2ccc(OC)cc2-c2cccc(O)c2)c(-c2cccc(O)c2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.58
RAB9A P51151 2/20 0.58
CYP1A2 P05177 4/20 0.55
CYP2C19 P33261 4/20 0.55
CYP3A4 P08684 4/20 0.55
HPGD P15428 3/20 0.55
LMNA P02545 2/20 0.55
PGR P06401 2/20 0.55
SLC6A2 P23975 2/20 0.55
ADORA3 P0DMS8 1/20 0.55
AR P10275 1/20 0.55
CHRM1 P11229 1/20 0.55
ALOX15 P16050 1/20 0.55
TBXA2R P21731 1/20 0.55
ADRA1A P35348 1/20 0.55
HIF1A Q16665 1/20 0.55
ALDH1A1 P00352 3/20 0.50
CYP2D6 P10635 3/20 0.50
MAPK1 P28482 2/20 0.50
PDE4A P27815 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31619636 0.90 SMN1; SMN2 (0.51) NPC1RAB9ACYP1A2CYP2C19CYP3A4
SCHEMBL8782870 0.84 CYP1A2 (0.57) NPC1RAB9ACYP1A2CYP2C19CYP3A4
SCHEMBL7532214 0.80 GSTP1 (0.62) NPC1RAB9ACYP1A2CYP2C19CYP3A4
SCHEMBL2934843 0.78 ALDH1A1 (0.56) NPC1RAB9ACYP1A2CYP2C19CYP3A4
SCHEMBL8202718 0.78 PRKAB2 (0.55) HPGDLMNAALDH1A1CYP2C8SMN1; SMN2
SCHEMBL2869177 0.78 TRIM24 (0.59) CYP1A2CYP2C19CYP3A4ARALDH1A1
SCHEMBL20208770 0.77 KDM4E (0.56) CYP1A2CYP2C19CYP3A4HPGDLMNA
SCHEMBL29706084 0.77 KDM4E (0.56) CYP1A2CYP2C19CYP3A4HPGDLMNA
SCHEMBL30739535 0.77 ALDH1A1 (0.68) NPC1RAB9ACYP1A2CYP2C19HPGD
SCHEMBL5144554 0.76 NPC1 (0.69) NPC1RAB9ACYP1A2CYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7767693-B2 Hsp90 family protein inhibitors KYOWA HAKKO KIRIN CO., LTD. (JP) 2010-08-03 US disclosed