SCHEMBL28699683

SCHEMBL28699683

COC(=O)CC(NC1(C)CCN(CCc2ccc3c(n2)N(C(=O)O)CCC3)C1)c1ccccc1

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 9/20 0.33
ITGB3 P05106 6/20 0.33
ITGB6 P18564 6/20 0.33
ITGB5 P18084 2/20 0.33
ITGB8 P26012 2/20 0.33
GRM7 Q14831 3/20 0.32
EPHX2 P34913 1/20 0.32
OPRM1 P35372 1/20 0.31
KCNH2 Q12809 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
FGFR4 P22455 3/20 0.31
ITGA2B P08514 1/20 0.31
CCR5 P51681 1/20 0.31
TACR3 P29371 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28984873 0.91 ATM (0.34) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL30474556 0.85 ITGAV (0.49) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL28692089 0.85 ITGAV (0.49) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL28708238 0.77 ITGB3 (0.57) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL28698397 0.74 ITGAV (0.41) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL20140491 0.73 ITGB3 (0.43) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL29369724 0.71 LMNA (0.40) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL3095932 0.71 FGFR4 (0.40) FGFR4
SCHEMBL28337910 0.70 ITGAV (0.40) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL29370042 0.70 ITGB3 (0.36) ITGAVITGB3ITGB6ITGB5ITGB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113354635-A Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2021-09-07 CN disclosed