SCHEMBL28698397

SCHEMBL28698397

COC(=O)CC(N[C@@H]1CCN(CCc2ccc3c(n2)N(C(=O)O)CCC3)C1)c1cccc(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 13/20 0.41
ITGB3 P05106 11/20 0.41
ITGB5 P18084 3/20 0.41
ITGB6 P18564 12/20 0.38
ITGB8 P26012 2/20 0.38
CCR5 P51681 1/20 0.36
ADRB1 P08588 1/20 0.34
ADRB3 P13945 1/20 0.34
HRH3 Q9Y5N1 2/20 0.34
WDR5 P61964 1/20 0.34
ITGB1 P05556 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28709236 0.91 ITGB3 (0.37) ITGAVITGB3ITGB5ITGB6ITGB8
SCHEMBL28685987 0.87 ITGAV (0.47) ITGAVITGB3ITGB5ITGB6ITGB8
SCHEMBL28699758 0.85 ITGAV (0.56) ITGAVITGB3ITGB5ITGB6ITGB8
SCHEMBL28699760 0.82 ITGAV (0.46) ITGAVITGB3ITGB5ITGB6ITGB8
SCHEMBL20140491 0.79 ITGB3 (0.43) ITGAVITGB3ITGB5ITGB6ITGB8
SCHEMBL28699748 0.78 ITGAV (0.35) ITGAVITGB3ITGB5ITGB6ITGB1
SCHEMBL28696946 0.76 CCR5 (0.39) ITGAVITGB3ITGB5ITGB6ITGB8
SCHEMBL28686054 0.76 WDR5 (0.42) WDR5
SCHEMBL27003291 0.75 ITGB3 (0.40) ITGAVITGB3ITGB5ITGB6ITGB8
SCHEMBL28699683 0.74 ITGAV (0.33) ITGAVITGB3ITGB5ITGB6ITGB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113354635-B Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2023-04-18 CN disclosed
CN-113354635-A Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2021-09-07 CN disclosed