SCHEMBL28699758

SCHEMBL28699758

COC(=O)CC(NC1CCN(CCc2ccc3c(n2)NCCC3)C1)c1cccc(Cl)c1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 20/20 0.56
ITGB3 P05106 17/20 0.56
ITGB5 P18084 8/20 0.56
ITGB6 P18564 16/20 0.54
ITGB8 P26012 5/20 0.54
ITGB1 P05556 3/20 0.47
KCNH2 Q12809 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28692096 0.86 ITGB3 (0.53) ITGAVITGB3ITGB5ITGB6ITGB8
SCHEMBL28698397 0.85 ITGAV (0.41) ITGAVITGB3ITGB5ITGB6ITGB8
SCHEMBL28701915 0.84 ITGB3 (0.56) ITGAVITGB3ITGB5ITGB6ITGB8
SCHEMBL28701920 0.84 ITGB3 (0.56) ITGAVITGB3ITGB5ITGB6ITGB8
SCHEMBL28709236 0.82 ITGB3 (0.37) ITGAVITGB3ITGB5ITGB6ITGB8
SCHEMBL28685968 0.80 ITGAV (0.68) ITGAVITGB3ITGB5ITGB6ITGB8
SCHEMBL28685964 0.80 ITGAV (0.68) ITGAVITGB3ITGB5ITGB6ITGB8
SCHEMBL30487545 0.78 ITGAV (0.60) ITGAVITGB3ITGB5ITGB6ITGB8
SCHEMBL28744348 0.78 ITGAV (0.60) ITGAVITGB3ITGB5ITGB6ITGB8
SCHEMBL20158342 0.78 ITGAV (0.60) ITGAVITGB3ITGB5ITGB6ITGB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113354635-B Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2023-04-18 CN disclosed
CN-113354635-A Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2021-09-07 CN disclosed