SCHEMBL28709236

SCHEMBL28709236

COC(=O)CC(N[C@@H]1CCN(CCc2ccc3c(n2)N(C(=O)OC(C)(C)C)CCC3)C1)c1cccc(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 10/20 0.37
ITGAV P06756 10/20 0.37
ITGB5 P18084 2/20 0.37
ITGB6 P18564 9/20 0.35
ITGB8 P26012 1/20 0.35
STS P08842 1/20 0.34
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34
CCR5 P51681 2/20 0.33
FNTA P49354 1/20 0.33
FNTB P49356 1/20 0.33
ADRB1 P08588 1/20 0.33
ADRB3 P13945 1/20 0.33
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28698397 0.91 ITGAV (0.41) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL28690115 0.82 ITGAV (0.48) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL28690112 0.82 ITGAV (0.48) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL28699758 0.82 ITGAV (0.56) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL29702194 0.80 ITGB3 (0.40) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL20158343 0.80 ITGB3 (0.40) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL28685987 0.79 ITGAV (0.47) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL28699743 0.78 STS (0.49) STSTP53MAPK1
SCHEMBL30474573 0.78 CCR5 (0.36) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL27406312 0.77 PRMT5 (0.39) ITGAVITGB6CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113354635-A Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2021-09-07 CN disclosed