SCHEMBL287022

SCHEMBL287022

Cc1ccc(N=C=Nc2ccc(C)cc2)cc1.Cc1ccccc1N=C=Nc1ccccc1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.43
CYP3A4 P08684 3/20 0.43
TDP1 Q9NUW8 2/20 0.43
TP53 P04637 1/20 0.43
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CYP2C9 P11712 1/20 0.36
TRPA1 O75762 1/20 0.36
POLB P06746 2/20 0.35
KMT2A Q03164 6/20 0.35
MEN1 O00255 4/20 0.35
L3MBTL1 Q9Y468 3/20 0.35
MAPT P10636 3/20 0.35
LMNA P02545 3/20 0.35
ALDH1A1 P00352 2/20 0.35
ACHE P22303 3/20 0.35
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2047233 0.94 TSHR (0.47) TSHRCYP3A4TDP1TP53MAPK1
SCHEMBL508210 0.88 MIF (0.43) TSHRCYP3A4TDP1TP53MAPK1
SCHEMBL8401752 0.88 MIF (0.43) TSHRCYP3A4TDP1TP53MAPK1
SCHEMBL437747 0.87 TSHR (0.47) TSHRCYP3A4TDP1TP53MAPK1
SCHEMBL29516244 0.87 TSHR (0.47) TSHRCYP3A4TDP1TP53MAPK1
SCHEMBL508209 0.83 MIF (0.46) TSHRTDP1MAPK1CYP2C9POLB
SCHEMBL159755 0.82 ACHE (0.47) TSHRTDP1MAPK1SMN1; SMN2CYP2C9
SCHEMBL14518105 0.78 CYP3A4 (0.51) TSHRCYP3A4TDP1TP53MAPK1
SCHEMBL12646532 0.77 FTO (0.46) TSHRCYP3A4TDP1TP53MAPK1
SCHEMBL9136636 0.77 TSHR (0.43) TSHRCYP3A4TDP1TP53MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427428-A1 O-IMINO-ISO-UREA COMPOUNDS AND POLYMERIZABLE COMPOSITIONS THEREOF BASF SE (DE) 2012-03-14 EP disclosed
WO-2010128062-A1 O-IMINO-ISO-UREA COMPOUNDS AND POLYMERIZABLE COMPOSITIONS THEREOF BASF SE (DE) 2010-11-11 WO disclosed
EP-0028683-A1 Antibiotic C-15003 PHO and production thereof Takeda Chemical Industries, Ltd. (JP) 1981-05-20 EP disclosed