SCHEMBL28703752

SCHEMBL28703752

COc1ccc(-c2csc(-c3csc(Nc4cc(Cl)cc(Cl)c4)n3)n2)cc1

nearest known ligand 0.80

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1B1 Q16678 12/20 0.80
CYP1A1 P04798 10/20 0.80
CYP1A2 P05177 9/20 0.72
ALOX5 P09917 3/20 0.70
PTGS2 P35354 3/20 0.67
MEN1 O00255 2/20 0.65
NPC1 O15118 2/20 0.65
GAA P10253 2/20 0.65
MAPT P10636 2/20 0.65
RAB9A P51151 2/20 0.65
KMT2A Q03164 2/20 0.65
SMN1; SMN2 Q16637 2/20 0.65
ALDH1A1 P00352 1/20 0.62
NFKB1 P19838 1/20 0.62
NFKB2 Q00653 1/20 0.62
RELA Q04206 1/20 0.62
MCL1 Q07820 1/20 0.62
VCP P55072 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29654197 0.90 CYP1B1 (0.74) CYP1B1CYP1A1CYP1A2ALOX5PTGS2
SCHEMBL28712406 0.90 CYP1B1 (0.74) CYP1B1CYP1A1CYP1A2ALOX5PTGS2
SCHEMBL28936901 0.89 ALOX5 (0.88) CYP1B1CYP1A1CYP1A2ALOX5PTGS2
SCHEMBL28701564 0.84 CYP1B1 (0.77) CYP1B1CYP1A1CYP1A2ALOX5NPC1
SCHEMBL28712378 0.84 CYP1A1 (1.00) CYP1B1CYP1A1CYP1A2ALOX5MEN1
SCHEMBL28720648 0.84 CYP1A1 (1.00) CYP1B1CYP1A1CYP1A2ALOX5VCP
SCHEMBL12297262 0.83 ALOX5 (1.00) ALOX5PTGS2MEN1NPC1GAA
SCHEMBL28720665 0.81 CYP1B1 (1.00) CYP1B1CYP1A1CYP1A2ALOX5MEN1
SCHEMBL7537503 0.81 PTGS2 (1.00) CYP1B1CYP1A1CYP1A2ALOX5PTGS2
SCHEMBL12297852 0.81 PTGS2 (1.00) CYP1B1CYP1A1CYP1A2ALOX5PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114249702-A N-aryl- [2,4 '-bithiazole ] -2' -amine compound and preparation and application thereof 沈阳药科大学 2022-03-29 CN disclosed