SCHEMBL28708441

SCHEMBL28708441

N#Cc1cc(F)cc(CN2CCNCC2)c1OCOC(=O)C1CC1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 1/20 0.43
ALDH1A1 P00352 6/20 0.39
TDP1 Q9NUW8 2/20 0.39
MLNR O43193 1/20 0.37
POLB P06746 1/20 0.34
KDM4E B2RXH2 2/20 0.33
CHRM3 P20309 1/20 0.33
CHRM4 P08173 2/20 0.32
CYP1A2 P05177 1/20 0.32
CHRM2 P08172 1/20 0.32
SLC6A4 P31645 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
CTSC P53634 1/20 0.32
APOBEC3A P31941 1/20 0.31
CTDSP1 Q9GZU7 1/20 0.31
APOBEC3G Q9HC16 1/20 0.31
GPR6 P46095 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28696633 0.83 MGLL (0.51) MGLLALDH1A1TDP1
SCHEMBL28714863 0.81 MGLL (0.69) MGLL
SCHEMBL20137015 0.77 MGLL (0.69) MGLLCHRM3
SCHEMBL28699391 0.71 ALDH1A1 (0.44) MGLLALDH1A1TDP1MLNRPOLB
SCHEMBL20137036 0.68 MGLL (0.68) MGLL
SCHEMBL20137140 0.67 MGLL (0.67) MGLL
SCHEMBL20167062 0.64 MGLL (0.63) MGLLALDH1A1POLBKDM4E
SCHEMBL21883706 0.63 MGLL (0.36) MGLLALDH1A1KDM4ECYP1A2
SCHEMBL28086944 0.62 SLC6A4 (0.43) ALDH1A1TDP1MLNRKDM4ECHRM3
SCHEMBL28887675 0.60 DDR1 (0.42) MGLLALDH1A1TDP1MLNRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110267963-B MAGL inhibitors H.隆德贝克有限公司 2022-04-01 CN disclosed