SCHEMBL2870864

SCHEMBL2870864

O=C(O)c1coc(-c2cccc(-c3ccccc3)c2)n1

nearest known ligand 0.74

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.74
HDAC8 Q9BY41 4/20 0.74
HDAC6 Q9UBN7 4/20 0.74
ALDH1A1 P00352 1/20 0.59
PDE4B Q07343 5/20 0.49
KMO O15229 2/20 0.49
PTPN1 P18031 2/20 0.49
PSMB8 P28062 1/20 0.46
ACMSD Q8TDX5 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2866244 0.88 HDAC1 (0.71) HDAC1HDAC8HDAC6ALDH1A1PDE4B
SCHEMBL287420 0.88 ALDH1A1 (0.74) HDAC1HDAC8HDAC6ALDH1A1PDE4B
SCHEMBL12522824 0.88 HDAC1 (0.58) HDAC1HDAC8HDAC6ALDH1A1PDE4B
SCHEMBL31558487 0.84 PDE4B (0.63) HDAC1HDAC8HDAC6ALDH1A1PDE4B
SCHEMBL2868465 0.84 ADRB2 (0.55) HDAC1HDAC8HDAC6ALDH1A1PDE4B
SCHEMBL12521272 0.83 HDAC1 (0.72) HDAC1HDAC8HDAC6ALDH1A1PDE4B
SCHEMBL2872214 0.82 HDAC1 (0.52) HDAC1HDAC8HDAC6ALDH1A1PDE4B
SCHEMBL12521298 0.81 HDAC1 (0.51) HDAC1HDAC8HDAC6ALDH1A1PDE4B
SCHEMBL2638386 0.81 ADRB2 (0.53) HDAC1HDAC8HDAC6ALDH1A1PDE4B
SCHEMBL31604686 0.81 KMO (0.54) HDAC1HDAC8HDAC6ALDH1A1PDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2307394-B1 SULPHONAMIDES AS VANILLOID RECEPTOR ANTAGONIST AMOREPACIFIC CORP (KR) 2012-09-26 EP disclosed
WO-2010002209-A2 NOVEL COMPOUNDS, ISOMER THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS VANILLOID RECEPTOR ANTAGONIST AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AMOREPACIFIC CORPORATION (KR) 2010-01-07 WO disclosed