SCHEMBL28708702

SCHEMBL28708702

CC(COC(N)=O)(C(S)S)C(N)c1ccc(CO)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.35
PPARA Q07869 1/20 0.35
EPHX2 P34913 1/20 0.33
LMNA P02545 3/20 0.33
HSD17B10 Q99714 1/20 0.33
CYP3A4 P08684 2/20 0.32
CYP1A2 P05177 2/20 0.32
CYP2D6 P10635 2/20 0.32
CYP2C9 P11712 1/20 0.32
NFKB1 P19838 1/20 0.32
CYP2C19 P33261 1/20 0.32
PKM P14618 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
F2 P00734 1/20 0.31
PMP22 Q01453 1/20 0.31
NLRP3 Q96P20 1/20 0.31
EPHX1 P07099 1/20 0.31
KIF11 P52732 2/20 0.30
ADRB2 P07550 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1936445 0.71 PPARG (0.43) PPARGPPARAEPHX2LMNACYP1A2
SCHEMBL3643384 0.67 PPARG (0.41) PPARGPPARAEPHX2LMNACYP3A4
SCHEMBL28966364 0.64 EPHX1 (0.42) PPARGPPARALMNACYP2C9NFKB1
SCHEMBL1934151 0.64 EPHX1 (0.42) PPARGPPARALMNACYP2C9NFKB1
SCHEMBL1934595 0.64 KMT2A (0.44) PPARGPPARALMNASMN1; SMN2
SCHEMBL16569006 0.63 PPARG (0.44) PPARGPPARAEPHX2LMNACYP3A4
SCHEMBL8139642 0.63 EPHX1 (0.43) PPARGPPARAF2EPHX1KIF11
SCHEMBL1526008 0.62 EPHX1 (0.70) LMNACYP2C9NFKB1SMN1; SMN2PMP22
SCHEMBL1936079 0.62 LMNA (0.55) LMNAHSD17B10CYP3A4SMN1; SMN2
SCHEMBL23533687 0.61 F2 (0.43) CYP1A2CYP2D6PKMSMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114191428-A Eribulin-based antibody-drug conjugates and methods of use 卫材研究发展管理有限公司 2022-03-18 CN disclosed