SCHEMBL28709403

SCHEMBL28709403

COC(=O)CCNc1cccc(-n2nc(C)cc2C)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 6/20 0.43
MAPT P10636 5/20 0.43
HPGD P15428 3/20 0.43
KAT6A Q92794 1/20 0.42
MAPK1 P28482 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
LMNA P02545 3/20 0.42
ALDH1A1 P00352 3/20 0.42
GAA P10253 2/20 0.42
HTT P42858 2/20 0.42
L3MBTL1 Q9Y468 3/20 0.41
TDP1 Q9NUW8 1/20 0.41
TSHR P16473 2/20 0.41
KCNJ6 P48051 1/20 0.40
KCNJ5 P48544 1/20 0.40
KCNJ3 P48549 1/20 0.40
NPY5R Q15761 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28709234 0.88 MAPT (0.47) SMN1; SMN2MAPTHPGDMAPK1MEN1
SCHEMBL16140804 0.78 MAPT (0.50) MAPTHPGDKAT6AKMT2AALDH1A1
SCHEMBL28709251 0.77 KAT6A (0.49) SMN1; SMN2MAPTHPGDKAT6AMAPK1
SCHEMBL9468482 0.75 MAPT (0.62) SMN1; SMN2MAPTHPGDMAPK1MEN1
SCHEMBL25624042 0.73 MAPT (0.44) SMN1; SMN2MAPTHPGDKAT6AMAPK1
SCHEMBL11702794 0.72 POLB (0.54) SMN1; SMN2MAPTMAPK1MEN1KMT2A
SCHEMBL18289071 0.72 GAA (0.62) SMN1; SMN2MAPTHPGDMAPK1MEN1
SCHEMBL10126717 0.71 MTNR1B (0.67) SMN1; SMN2HPGDKMT2AALDH1A1GAA
SCHEMBL16793988 0.71 SMN1; SMN2 (0.52) SMN1; SMN2MAPTHPGDMEN1KMT2A
SCHEMBL28690119 0.70 MAPT (0.47) SMN1; SMN2MAPTHPGDKAT6AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113354635-B Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2023-04-18 CN disclosed
CN-113354635-A Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2021-09-07 CN disclosed