SCHEMBL28722018

SCHEMBL28722018

FC(F)(F)c1ccc2cccnc2c1Br

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.52
CCR1 P32246 3/20 0.52
CCR5 P51681 3/20 0.52
CCR8 P51685 3/20 0.52
MMP2 P08253 2/20 0.52
TSHR P16473 2/20 0.52
HTT P42858 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
KDM4E B2RXH2 1/20 0.52
GMNN O75496 1/20 0.52
TP53 P04637 1/20 0.52
HSP90AA1 P07900 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
MAPT P10636 1/20 0.52
MMP9 P14780 1/20 0.52
ALOX15 P16050 1/20 0.52
NFKB1 P19838 1/20 0.52
MMP8 P22894 1/20 0.52
THPO P40225 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29496277 1.00 LMNA (0.52) LMNACCR1CCR5CCR8MMP2
SCHEMBL22016210 0.79 CCR1 (0.52) LMNACCR1CCR5CCR8MMP2
SCHEMBL2569765 0.77 PSMD14 (0.55) LMNACCR1CCR5CCR8MMP2
SCHEMBL29935933 0.77 PSMD14 (0.55) LMNACCR1CCR5CCR8MMP2
SCHEMBL24312088 0.76 LMNA (0.48) LMNACCR1CCR5CCR8MMP2
SCHEMBL31716531 0.76 LMNA (0.58) LMNACCR1CCR5CCR8MMP2
SCHEMBL28845889 0.75 TOP1 (0.48) LMNACCR1CCR5CCR8MMP2
SCHEMBL17940499 0.75 KDM4E (0.47) LMNACCR1CCR5CCR8MMP2
SCHEMBL20392639 0.74 PSMD14 (0.41) LMNACCR1CCR5CCR8MMP2
Phenanthroline SCHEMBL12478422 0.72 CCR1 (0.73) LMNACCR1CCR5CCR8MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114269730-A 5-heteroaryl-pyridin-2-amine compounds as neuropeptide FF receptor antagonists 多曼治疗学公司 2022-04-01 CN disclosed