SCHEMBL28724728

SCHEMBL28724728

COS(=O)(=O)Cc1cc(F)c(C#N)cc1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 2/20 0.40
TUBB4A P04350 1/20 0.32
TUBB P07437 1/20 0.32
TUBA3C P0DPH7 1/20 0.32
STAT3 P40763 1/20 0.32
TUBA1B P68363 1/20 0.32
TUBA4A P68366 1/20 0.32
TUBB4B P68371 1/20 0.32
TUBB3 Q13509 1/20 0.32
TUBB2A Q13885 1/20 0.32
TUBB8 Q3ZCM7 1/20 0.32
TUBA3E Q6PEY2 1/20 0.32
TUBA1A Q71U36 1/20 0.32
TUBA1C Q9BQE3 1/20 0.32
TUBB6 Q9BUF5 1/20 0.32
TUBB2B Q9BVA1 1/20 0.32
TUBB1 Q9H4B7 1/20 0.32
BRD4 O60885 1/20 0.32
CYP11B1 P15538 2/20 0.31
CYP11B2 P19099 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13766377 0.76 TRPV4 (0.50) TRPV4CYP11B1CYP11B2
SCHEMBL3149348 0.75 TRPV4 (0.40) TRPV4SLC22A12
SCHEMBL18215048 0.75 TRPV4 (0.46) TRPV4CYP11B1CYP11B2
SCHEMBL30154484 0.72 MAPT (0.40) TRPV4
SCHEMBL23832263 0.72 MAPT (0.40) TRPV4
SCHEMBL29183220 0.71 HTR2A (0.35)
SCHEMBL29183259 0.71 ALDH1A1 (0.30)
SCHEMBL30184743 0.71 ALDH1A1 (0.30)
SCHEMBL28724729 0.70 TRPV4 (0.41) TRPV4CYP11B1CYP11B2SLC22A12
SCHEMBL363766 0.69 TRPV4 (0.50) TRPV4CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114364672-A Benzisoxazole sulfonamide derivatives 辉瑞大药厂 2022-04-15 CN disclosed