SCHEMBL28742010

SCHEMBL28742010

O=C(CCC(=O)NC1CCN(Cc2ccccc2)CC1)NNc1ccc(Cl)nn1

nearest known ligand 0.59

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 17/20 0.59
SLC6A12 P48065 1/20 0.54
POLB P06746 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29640453 1.00 SIGMAR1 (0.59) SIGMAR1SLC6A12POLB
SCHEMBL22966087 0.82 SIGMAR1 (0.62) SIGMAR1POLB
SCHEMBL28741993 0.79 SIGMAR1 (0.77) SIGMAR1POLB
SCHEMBL2821246 0.78 ACHE (0.73) SIGMAR1SLC6A12
SCHEMBL6333442 0.77 SIGMAR1 (0.73) SIGMAR1POLB
SCHEMBL4848450 0.77 SIGMAR1 (0.77) SIGMAR1POLB
SCHEMBL22966100 0.76 OPRM1 (0.41) SIGMAR1SLC6A12
SCHEMBL13360982 0.76 SIGMAR1 (0.75) SIGMAR1POLB
SCHEMBL9852459 0.76 SIGMAR1 (0.75) SIGMAR1POLB
SCHEMBL5862113 0.75 SIGMAR1 (1.00) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114450006-A TrkB positive allosteric modulators 斯特拉斯堡大学 2022-05-06 CN disclosed