SCHEMBL28746480

SCHEMBL28746480

CCOC(=O)c1cc2cc(NC(=O)[C@H](Cc3ccc(NC(=O)C(C)C)cc3)NC(=O)OC(C)(C)C)ccc2[nH]1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 4/20 0.53
MMP2 P08253 3/20 0.47
F11 P03951 9/20 0.47
HDAC8 Q9BY41 1/20 0.47
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 2/20 0.44
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
LEF1 Q9UJU2 1/20 0.43
NPC1 O15118 1/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
HRH3 Q9Y5N1 1/20 0.42
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
MMP14 P50281 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28746481 1.00 MMP13 (0.53) MMP13MMP2F11HDAC8KDM4E
SCHEMBL28746519 0.92 MMP13 (0.50) MMP13MMP2F11HDAC8KDM4E
SCHEMBL28292652 0.92 MMP13 (0.53) MMP13MMP2F11HDAC8KDM4E
SCHEMBL23466599 0.92 MMP13 (0.55) MMP13MMP2F11HDAC8KDM4E
SCHEMBL23466603 0.92 MMP13 (0.55) MMP13MMP2F11HDAC8KDM4E
SCHEMBL29758100 0.92 MMP13 (0.55) MMP13MMP2F11HDAC8KDM4E
SCHEMBL28746504 0.90 MMP13 (0.52) MMP13MMP2F11HDAC8KDM4E
SCHEMBL28746506 0.90 MMP13 (0.52) MMP13MMP2F11HDAC8KDM4E
SCHEMBL28941305 0.90 F11 (0.51) MMP13MMP2F11HDAC8KDM4E
SCHEMBL28941304 0.90 F11 (0.51) MMP13MMP2F11HDAC8KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114539158-A FXIa inhibitor compound and preparation method and application thereof 沈阳药科大学 2022-05-27 CN disclosed