SCHEMBL2875249

SCHEMBL2875249

Cc1cc(NNc2cc(C)cc(C3CCc4ccccc4C3)n2)nc(C2=Cc3ccccc3CC2)c1

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TRPV3 Q8NET8 1/20 0.34
CYP19A1 P11511 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
NISCH Q9Y2I1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2875248 0.84 GRIN2D (0.38) TRPV3CYP19A1CYP11B1CYP11B2NISCH
SCHEMBL2087271 0.70 GRIN2D (0.46) TRPV3
SCHEMBL2090630 0.70 GRIN2D (0.46) CYP19A1CYP11B1CYP11B2NISCH
SCHEMBL5865169 0.69 CYP19A1 (0.35) CYP19A1CYP11B1CYP11B2NISCH
SCHEMBL5865222 0.64 CYP11B1 (0.42) CYP19A1CYP11B1CYP11B2NISCH
SCHEMBL5865518 0.63 GRIN2D (0.43) CYP19A1CYP11B1CYP11B2NISCH
Fumaric Acid SCHEMBL5865172 0.62 GRIN2D (0.39) CYP19A1CYP11B1CYP11B2NISCH
Fumaric Acid SCHEMBL5865164 0.62 GRIN2D (0.39) CYP19A1CYP11B1CYP11B2NISCH
SCHEMBL24266487 0.62 TRPV3 (0.43) TRPV3
SCHEMBL5607529 0.60 CYP11B2 (0.57) CYP19A1CYP11B1CYP11B2NISCH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2227452-A2 PYRIDINE COMPOUNDS F. Hoffmann-La Roche AG (CH) 2010-09-15 EP disclosed
WO-2009068468-A2 PYRIDINE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2009-06-04 WO disclosed