SCHEMBL287526

SCHEMBL287526

CCOC(=O)c1ccccc1NC(=O)C1C=CN(CC(=O)c2cccs2)C=C1

nearest known ligand 0.61

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.61
ALDH1A1 P00352 7/20 0.51
KMT2A Q03164 4/20 0.51
MEN1 O00255 3/20 0.51
RAB9A P51151 1/20 0.51
NPSR1 Q6W5P4 3/20 0.44
TP53 P04637 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
HTT P42858 1/20 0.44
CNR2 P34972 1/20 0.44
KDM4E B2RXH2 5/20 0.43
HSD17B10 Q99714 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
HPGD P15428 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL287235 0.79 TSHR (0.63) TSHRALDH1A1KMT2AMEN1RAB9A
SCHEMBL287525 0.73 ALDH1A1 (0.50) TSHRALDH1A1RAB9ANPSR1TDP1
SCHEMBL9767800 0.68 ALDH1A1 (0.67) TSHRALDH1A1KMT2AMEN1RAB9A
SCHEMBL2860044 0.66 KDM4E (0.68) TSHRALDH1A1KMT2AMEN1NPSR1
SCHEMBL10501732 0.66 KDM4E (0.78) TSHRALDH1A1KMT2ANPSR1TP53
SCHEMBL7312805 0.66 LMNA (0.71) TSHRALDH1A1NPSR1TP53TDP1
SCHEMBL31126834 0.66 KDM4E (0.68) TSHRALDH1A1KMT2AMEN1NPSR1
SCHEMBL10438008 0.66 KDM4E (0.68) TSHRALDH1A1RAB9ANPSR1TP53
SCHEMBL422787 0.65 RAB9A (0.62) TSHRALDH1A1KMT2AMEN1RAB9A
SCHEMBL14085807 0.65 KDM4E (0.76) TSHRALDH1A1KMT2ANPSR1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427432-A2 NOVEL HETEROCYCLIC COMPOUNDS Torrent Pharmaceuticals Limited (IN) 2012-03-14 EP disclosed
WO-2010128528-A2 NOVEL HETEROCYCLIC COMPOUNDS TORRENT PHARMACEUTICALS LIMITED (IN) 2010-11-11 WO disclosed