SCHEMBL28758652

SCHEMBL28758652

CC(=O)OCCc1nc(N2CCN(C)CC2)ccc1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.41
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 3/20 0.41
CYP2C19 P33261 2/20 0.41
TSHR P16473 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
HRH4 Q9H3N8 3/20 0.40
HRH3 Q9Y5N1 3/20 0.40
PTK2 Q05397 5/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
PARP1 P09874 1/20 0.39
HPGD P15428 1/20 0.38
ADRB2 P07550 1/20 0.38
UCHL3 P15374 1/20 0.37
TACR1 P25103 2/20 0.37
HTR3E A5X5Y0 1/20 0.36
HTR3B O95264 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3238492 0.81 SMN1; SMN2 (0.45) CYP1A2KDM4EALDH1A1CYP2C19TSHR
SCHEMBL856329 0.80 PTK2 (0.47) CYP1A2KDM4EALDH1A1CYP2C19TSHR
SCHEMBL27627608 0.75 NOTUM (0.39) KDM4EALDH1A1SMN1; SMN2
SCHEMBL27563803 0.74 HTR3A (0.54) KDM4EALDH1A1HRH3HTR3A
SCHEMBL28758653 0.74 CYP1A2 (0.41) CYP1A2KDM4EALDH1A1CYP2C19TSHR
SCHEMBL860986 0.74 SMN1; SMN2 (0.45) CYP1A2KDM4EALDH1A1CYP2C19TSHR
SCHEMBL1433676 0.69 AOC3 (0.68) PTK2
Hydrochloric Acid SCHEMBL1432850 0.68 AOC3 (0.67) PTK2
SCHEMBL19012355 0.67 HRH4 (0.46) CYP1A2KDM4EALDH1A1CYP2C19TSHR
SCHEMBL24190079 0.66 CYP1A2 (0.47) CYP1A2KDM4EALDH1A1CYP2C19TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100439359-C Indolylmaleimide derivatives NOVARTIS AG (CH) 2008-12-03 CN disclosed
CN-1742005-A Indolylmaleimide derivatives NOVARTIS AG (CH) 2006-03-01 CN disclosed