SCHEMBL28758653

SCHEMBL28758653

CC(=O)OC(C)c1nc(N2CCN(C)CC2)ccc1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.41
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 3/20 0.41
CYP2C19 P33261 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
DRD2 P14416 3/20 0.39
HTR6 P50406 3/20 0.39
HTR1A P08908 2/20 0.39
HTR2A P28223 2/20 0.39
HTR7 P34969 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PARP1 P09874 1/20 0.39
TACR1 P25103 2/20 0.38
HRH4 Q9H3N8 4/20 0.38
HRH3 Q9Y5N1 3/20 0.38
UCHL3 P15374 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL860986 0.78 SMN1; SMN2 (0.45) CYP1A2KDM4EALDH1A1CYP2C19CYP3A4
SCHEMBL27627609 0.75 ABHD6 (0.34) KDM4E
SCHEMBL28758652 0.74 CYP1A2 (0.41) CYP1A2KDM4EALDH1A1CYP2C19CYP3A4
SCHEMBL856329 0.70 PTK2 (0.47) CYP1A2KDM4EALDH1A1CYP2C19CYP3A4
SCHEMBL3238492 0.69 SMN1; SMN2 (0.45) CYP1A2KDM4EALDH1A1CYP2C19CYP3A4
SCHEMBL11991745 0.67 CNR2 (0.47) KDM4EADRB2
SCHEMBL19012355 0.67 HRH4 (0.46) CYP1A2KDM4EALDH1A1CYP2C19CYP3A4
SCHEMBL24190079 0.66 CYP1A2 (0.47) CYP1A2KDM4EALDH1A1CYP2C19CYP3A4
SCHEMBL1432175 0.65 ADRB2 (0.59) SMN1; SMN2ADRB2
SCHEMBL29676150 0.65 NPC1 (0.44) KDM4EALDH1A1PARP1HRH4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100439359-C Indolylmaleimide derivatives NOVARTIS AG (CH) 2008-12-03 CN disclosed
CN-1742005-A Indolylmaleimide derivatives NOVARTIS AG (CH) 2006-03-01 CN disclosed