SCHEMBL28764512

SCHEMBL28764512

CC(C)(C)CC(C(=O)NN)c1cccs1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.40
GLS O94925 1/20 0.38
CTSC P53634 2/20 0.38
HDAC2 Q92769 5/20 0.37
HDAC1 Q13547 4/20 0.37
HDAC3 O15379 2/20 0.37
TSHR P16473 2/20 0.37
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
KEAP1 Q14145 1/20 0.36
TP53 P04637 2/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27680341 0.78 HTT (0.44) ALOX5GLSHDAC1HDAC3TSHR
SCHEMBL27756817 0.72 ALOX5 (0.37) ALOX5GLSTSHRTP53MAPT
SCHEMBL6614649 0.71 ALOX5 (0.42) ALOX5GLSHDAC2HDAC1HDAC3
SCHEMBL20993292 0.71 ALOX5 (0.38) ALOX5CTSCTSHRCES2CES1
SCHEMBL17829522 0.71 NPC1 (0.43) ALOX5TSHRCES2CES1KEAP1
SCHEMBL6464486 0.68 ALOX5 (0.50) ALOX5GLSTSHRCES2CES1
SCHEMBL10210730 0.68 ALOX5 (0.50) ALOX5GLSTSHRCES2CES1
SCHEMBL20899846 0.68 GAA (0.42) ALOX5GLSTSHRCES2CES1
SCHEMBL7605356 0.67 MAPT (0.47) ALOX5TSHRMAPTRAB9A
SCHEMBL7411580 0.67 MAPT (0.47) ALOX5TSHRMAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101014578-B Triazole derivative or salt thereof ASTELLAS PHARMA INC 2011-01-19 CN disclosed
CN-101014578-A Triazole derivative or salt thereof ASTELLAS PHARMA INC (JP) 2007-08-08 CN disclosed