SCHEMBL28769596

SCHEMBL28769596

C=Cc1c(CCCC)ccnc1Cl

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTRC Q99895 1/20 0.36
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
THRA P10827 2/20 0.32
THRB P10828 2/20 0.32
ALDH1A1 P00352 1/20 0.32
HTT P42858 1/20 0.32
TYR P14679 1/20 0.32
CCNB2 O95067 1/20 0.31
CDK1 P06493 1/20 0.31
CCNB1 P14635 1/20 0.31
GSK3A P49840 1/20 0.31
GSK3B P49841 1/20 0.31
CCNB3 Q8WWL7 1/20 0.31
TLR8 Q9NR97 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15696056 0.78 TLR8 (0.33) HTR2AHTR2CHTR2BMEN1KMT2A
SCHEMBL28124885 0.77 CTRC (0.39) CTRCHTR2AHTR2CHTR2BTYR
SCHEMBL27777055 0.76 CTRC (0.41) CTRCHTR2AHTR2CHTR2BMEN1
SCHEMBL27857665 0.74 CTRC (0.37) CTRCHTR2AHTR2CHTR2BHTT
SCHEMBL22791948 0.72 LIPG (0.40) CTRCHTR2AHTR2CHTR2BMEN1
SCHEMBL12802233 0.72 CYP3A4 (0.42) THRATHRBTYR
SCHEMBL27754223 0.72 ALDH1A1 (0.41) CTRCKMT2AALDH1A1HTT
SCHEMBL1704724 0.72 CTRC (0.40) CTRCALDH1A1TLR8
SCHEMBL16828251 0.71 TYR (0.38) CTRCHTR2AHTR2CHTR2BMEN1
SCHEMBL19310672 0.71 TDP1 (0.35) CTRCHTR2AHTR2CHTR2BMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101160285-A Substituted sulfonylaminoarylmethyl cyclopropanecarboxamide as vr1 receptor antagonists PFIZER (US) 2008-04-09 CN disclosed