Thiophene

Thiophene

SCHEMBL28772829

O=C(O)c1ccc([N+](=O)[O-])cc1O.c1ccsc1

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.55
TDP1 Q9NUW8 2/20 0.55
CYP3A4 P08684 2/20 0.55
ALOX15 P16050 1/20 0.55
GPR35 Q9HC97 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.48
CTSV O60911 1/20 0.48
CTSL P07711 1/20 0.48
MAPT P10636 4/20 0.48
TP53 P04637 2/20 0.46
GAA P10253 2/20 0.46
ESR2 Q92731 1/20 0.46
KDM4E B2RXH2 1/20 0.46
PTPN1 P18031 1/20 0.46
CXCR1 P25024 1/20 0.46
CXCR2 P25025 1/20 0.46
KCNMA1 Q12791 1/20 0.46
CES2 O00748 1/20 0.46
AKR1C4 P17516 1/20 0.45
AKR1C3 P42330 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL578933 0.90 ALDH1A1 (0.66) ALDH1A1TDP1CYP3A4ALOX15GPR35
SCHEMBL28281676 0.89 ALDH1A1 (0.64) ALDH1A1TDP1CYP3A4ALOX15GPR35
SCHEMBL10082315 0.80 ALDH1A1 (0.54) ALDH1A1TDP1CYP3A4ALOX15GPR35
SCHEMBL6850686 0.78 HNF4A (0.64) ALDH1A1TDP1CYP3A4ALOX15SMN1; SMN2
Thiophene SCHEMBL27870135 0.77 KDM4E (0.52) ALDH1A1TDP1CYP3A4SMN1; SMN2MAPT
SCHEMBL129889 0.76 ALDH1A1 (0.69) ALDH1A1TDP1CYP3A4ALOX15GPR35
SCHEMBL30322798 0.76 ALDH1A1 (0.69) ALDH1A1TDP1CYP3A4ALOX15GPR35
SCHEMBL27497022 0.76 GAA (0.60) ALDH1A1GPR35SMN1; SMN2MAPTTP53
Benzoic Acid SCHEMBL28487710 0.76 SRD5A2 (0.57) ALDH1A1TDP1CYP3A4ALOX15SMN1; SMN2
SCHEMBL260006 0.76 ALDH1A1 (0.70) ALDH1A1TDP1CYP3A4ALOX15SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101088997-A Improved process of preparing Raltitrexed XIUHUA WEI (CN) 2007-12-19 CN claimed
CN-101088997-A Improved process of preparing Raltitrexed XIUHUA WEI (CN) 2007-12-19 CN disclosed