SCHEMBL28774604

SCHEMBL28774604

C=C(C(=O)O)c1ccc(Br)s1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.63
CES2 O00748 1/20 0.59
CES1 P23141 1/20 0.59
GSK3B P49841 2/20 0.52
KMT2A Q03164 5/20 0.49
ALDH1A1 P00352 4/20 0.49
HPGD P15428 2/20 0.46
POLB P06746 2/20 0.46
GAA P10253 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
KDM4E B2RXH2 2/20 0.44
ESR1 P03372 1/20 0.44
MEN1 O00255 2/20 0.42
NPC1 O15118 4/20 0.39
RAB9A P51151 4/20 0.39
TGM2 P21980 1/20 0.39
TGM1 P22735 1/20 0.39
MITF O75030 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28774611 0.82 CES2 (0.57) DAOCES2CES1GSK3BKMT2A
SCHEMBL2820847 0.78 CES2 (0.78) DAOCES2CES1GSK3BKMT2A
SCHEMBL71972 0.78
SCHEMBL23959941 0.76 GSK3B (0.58) DAOCES2CES1GSK3BKMT2A
SCHEMBL27713496 0.75 DAO (0.63) DAOGSK3BKMT2AALDH1A1HPGD
SCHEMBL1244072 0.75 CES2 (0.73) DAOCES2CES1GSK3BKMT2A
SCHEMBL2508391 0.75 CES2 (0.58) DAOCES2CES1GSK3BKMT2A
SCHEMBL10915819 0.72 DAO (0.59) DAOCES2CES1GSK3BKMT2A
SCHEMBL1476181 0.71
SCHEMBL345568 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114573502-B Pleuromutilin aromatic heterocyclic acrylate compound, and synthetic method and application thereof 西安康远晟生物医药科技有限公司 2024-05-03 CN disclosed
CN-114573502-A Pleuromutilin aromatic heterocyclic acrylate compounds and synthesis method and application thereof 西安康远晟生物医药科技有限公司 2022-06-03 CN disclosed