SCHEMBL1244072

SCHEMBL1244072

O=C(c1ccc(Br)s1)c1ccc(Br)s1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.73
CES1 P23141 1/20 0.73
DAO P14920 1/20 0.70
KMT2A Q03164 6/20 0.62
ALDH1A1 P00352 4/20 0.62
GSK3B P49841 2/20 0.61
HPGD P15428 2/20 0.53
POLB P06746 2/20 0.53
GAA P10253 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
RXFP1 Q9HBX9 1/20 0.53
KDM4E B2RXH2 2/20 0.52
ESR1 P03372 1/20 0.52
NPC1 O15118 4/20 0.49
RAB9A P51151 4/20 0.49
MEN1 O00255 3/20 0.49
HCRTR1 O43613 1/20 0.49
MAPT P10636 1/20 0.49
TSHR P16473 1/20 0.49
CASP1 P29466 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2010106 0.83 ALDH1A1 (0.66) CES2CES1DAOKMT2AALDH1A1
SCHEMBL2008426 0.83 CES2 (0.57) CES2CES1DAOKMT2AALDH1A1
SCHEMBL71972 0.82
SCHEMBL29171652 0.81 CES2 (0.61) CES2CES1DAOKMT2AALDH1A1
SCHEMBL1476181 0.80
SCHEMBL345568 0.80
SCHEMBL1455897 0.80
SCHEMBL15891223 0.80 CES2 (0.53) CES2CES1DAOKMT2AALDH1A1
SCHEMBL8308134 0.80 DAO (0.57) CES2CES1DAOKMT2AALDH1A1
SCHEMBL15988673 0.78 GSK3B (0.73) CES2CES1DAOKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100343256-C Biaryl substituted diazabicycloalkane amides as nicotinic acetylcholine agonists ASTRAZENECA AB (SE) 2007-10-17 CN claimed
CN-1678615-A Biaryl substituted diazabicycloalkanes as nicotinic acetylcholine antagonists ASTRAZENECA AB (SE) 2005-10-05 CN claimed
CN-102460758-A Semiconductor compound and device comprising the same UNIV KENTUCKY RES FOUND 2012-05-16 CN disclosed
CN-102209540-A Treatment with alpha a7-selective ligands TARGACEPT INC 2011-10-05 CN disclosed
US-20110039841-A1 Novel compounds, their preparation and use NOVO NORDISK A/S (DK) 2011-02-17 US disclosed
EP-1763511-B1 PHENOXYACETIC ACID DERIVATIVES AS PPAR AGONISTS HIGH POINT PHARMACEUTICALS LLC (US) 2010-07-28 EP disclosed
CN-101056873-A Carbonyl-functionalized thiophene compounds and related device structures UNIV NORTHWESTERN (US) 2007-10-17 CN disclosed
CN-100343256-C Biaryl substituted diazabicycloalkane amides as nicotinic acetylcholine agonists ASTRAZENECA AB (SE) 2007-10-17 CN disclosed
EP-1763511-A1 PHENOXYACETIC ACID DERIVATIVES AS PPAR AGONISTS NOVO NORDISK A/S (DK) 2007-03-21 EP disclosed
WO-2005105735-A1 PHENOXYACETIC ACID DERIVATIVES AS PPAR AGONISTS NOVO NORDISK A/S (DK) 2005-11-10 WO disclosed
CN-1678615-A Biaryl substituted diazabicycloalkanes as nicotinic acetylcholine antagonists ASTRAZENECA AB (SE) 2005-10-05 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110039841-A1 Novel compounds, their preparation and use PPARG, PPARD, PPARA CES2 1343/4885CES1 188/4885DAO 4142/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.