SCHEMBL28775136

SCHEMBL28775136

C[C@H]1CN(C(=O)C(NC(=O)OC(C)(C)C)C2CCCCC2)CCN1C(=O)OCc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.54
PDK2 Q15119 1/20 0.54
PDK3 Q15120 1/20 0.54
PDK4 Q16654 1/20 0.54
CTSL P07711 1/20 0.54
ITGB3 P05106 1/20 0.47
ITGA2B P08514 1/20 0.47
IDH1 O75874 1/20 0.42
PDE4B Q07343 1/20 0.42
PARP1 P09874 1/20 0.42
PREP P48147 2/20 0.41
MAPK1 P28482 1/20 0.41
P2RX7 Q99572 2/20 0.41
SPR P35270 1/20 0.41
FKBP1A P62942 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28775133 1.00 PDK1 (0.54) PDK1PDK2PDK3PDK4CTSL
SCHEMBL28775139 1.00 PDK1 (0.54) PDK1PDK2PDK3PDK4CTSL
SCHEMBL28532691 0.93 CTSL (0.54) PDK1PDK2PDK3PDK4CTSL
SCHEMBL28532689 0.93 CTSL (0.54) PDK1PDK2PDK3PDK4CTSL
SCHEMBL28533147 0.88 CTSL (0.59) CTSLITGB3ITGA2BPDE4BMAPK1
SCHEMBL29715729 0.88 CTSL (0.59) CTSLITGB3ITGA2BPDE4BMAPK1
SCHEMBL29808694 0.87 PDK1 (0.48) PDK1PDK2PDK3PDK4CTSL
SCHEMBL523864 0.85 PDK1 (0.57) PDK1PDK2PDK3PDK4CTSL
SCHEMBL523865 0.85 PDK1 (0.57) PDK1PDK2PDK3PDK4CTSL
SCHEMBL2441255 0.84 CTSL (0.57) CTSLITGB3ITGA2BPREPFKBP1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114729004-A Heterocyclic compounds 日商泛美克斯股份有限公司 2022-07-08 CN disclosed