SCHEMBL28781978

SCHEMBL28781978

O=C(NC(=O)C(Cl)(Cl)Cl)Nc1c(C(=O)O)cnc(-c2cccc3cccc(Cl)c23)c1F

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KRAS P01116 12/20 0.36
HSD17B10 Q99714 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TSHR P16473 1/20 0.36
KMT2A Q03164 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
KMO O15229 2/20 0.34
CNR1 P21554 1/20 0.33
EPAS1 Q99814 1/20 0.33
DHODH Q02127 1/20 0.32
HAVCR2 Q8TDQ0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29921963 0.90 NPC1 (0.37) KRASKDM4EALDH1A1
SCHEMBL23043008 0.90 NPC1 (0.37) KRASKDM4EALDH1A1
SCHEMBL31497664 0.77 KEAP1 (0.32) KDM4EALDH1A1DHODH
SCHEMBL26965094 0.76 HAVCR2 (0.49) KRASHSD17B10KDM4EMEN1ALDH1A1
SCHEMBL29121526 0.74 MAPT (0.44) KDM4EMEN1ALDH1A1KMT2A
SCHEMBL26708861 0.70 AURKB (0.40) KDM4EMEN1ALDH1A1TSHRKMT2A
SCHEMBL29680567 0.68 NR4A2 (0.40) KRASKDM4E
SCHEMBL23043368 0.68 NR4A2 (0.40) KRASKDM4E
SCHEMBL28782012 0.67 KRAS (0.38) KRAS
SCHEMBL22208213 0.66 KDM4E (0.35) HSD17B10KDM4EMEN1ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114615981-A KRAS G12D inhibitors 米拉蒂治疗股份有限公司 2022-06-10 CN disclosed