SCHEMBL29921963

SCHEMBL29921963

COC(=O)c1cnc(-c2cccc3cccc(Cl)c23)c(F)c1NC(=O)NC(=O)C(Cl)(Cl)Cl

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPK1 P28482 1/20 0.37
KRAS P01116 16/20 0.35
NR4A2 P43354 1/20 0.34
PDK1 Q15118 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33
POLB P06746 1/20 0.32
PKM P14618 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23043008 1.00 NPC1 (0.37) NPC1KDM4EALDH1A1MAPK1KRAS
SCHEMBL28781978 0.90 KRAS (0.36) KDM4EALDH1A1KRAS
SCHEMBL29121526 0.79 MAPT (0.44) NPC1KDM4EALDH1A1POLBPKM
SCHEMBL29680567 0.78 NR4A2 (0.40) KDM4EKRASNR4A2
SCHEMBL23043368 0.78 NR4A2 (0.40) KDM4EKRASNR4A2
SCHEMBL31442170 0.78 ATR (0.37) NPC1KDM4EALDH1A1MAPK1PDK1
SCHEMBL26708861 0.78 AURKB (0.40) KDM4EALDH1A1MAPK1POLB
SCHEMBL28782012 0.76 KRAS (0.38) KRAS
SCHEMBL22208213 0.71 KDM4E (0.35) KDM4EALDH1A1MAPK1RAB9A
SCHEMBL30064964 0.71 KDM4E (0.35) KDM4EALDH1A1MAPK1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025053850-A1 COVALENT KRAS-BINDING COMPOUNDS FOR MEDICAL TREATMENT HYKU BIOSCIENCES INC. (US) 2025-03-13 WO disclosed
WO-2022187688-A1 COVALENT KRAS-BINDING COMPOUNDS FOR THERAPEUTIC PURPOSES UMBRA THERAPEUTICS INC. (US) 2022-09-09 WO disclosed