SCHEMBL28782811

SCHEMBL28782811

CC(C)(C#N)c1ccc(CN)c(CN)c1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SCN10A Q9Y5Y9 1/20 0.37
CYP19A1 P11511 1/20 0.33
UGT1A4 P22310 1/20 0.33
PDE4D Q08499 1/20 0.33
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
HTR1D P28221 1/20 0.31
KLF10 Q13118 1/20 0.31
RORC P51449 1/20 0.30
JAK2 O60674 1/20 0.30
ROCK2 O75116 1/20 0.30
PRKCQ Q04759 1/20 0.30
PRKCD Q05655 1/20 0.30
ROCK1 Q13464 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL307936 0.87 SCN10A (0.36) SCN10ACYP19A1UGT1A4PDE4DCNR1
SCHEMBL27755359 0.84 SCN10A (0.35) SCN10ACYP19A1UGT1A4PDE4DCNR1
SCHEMBL27755272 0.80 SCN10A (0.40) SCN10A
SCHEMBL27775906 0.79 DHODH (0.36) SCN10ARORCJAK2
SCHEMBL3944519 0.77 TAAR1 (0.43) SCN10AHTR1D
SCHEMBL309341 0.75 LOXL2 (0.48) CYP19A1UGT1A4PDE4DESR1ESR2
Hydrochloric Acid SCHEMBL3125965 0.73 LOXL2 (0.47) ESR1ESR2RORC
SCHEMBL6563317 0.72 KIF11 (0.41) SCN10ACYP19A1UGT1A4PDE4DESR1
SCHEMBL18560992 0.71 KLF10 (0.43) SCN10ACNR1CNR2ESR1ESR2
SCHEMBL17157402 0.71 ESR1 (0.36) SCN10ACYP19A1UGT1A4PDE4DESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101792436-A Benzimidazole derivatives used in the treatment of diseases associated with vanilloid receptor 1 ASTRAZENECA R & D SODERTALJE 2010-08-04 CN disclosed
CN-101522637-A Benzimidazole derivatives useful for the treatment of vanilloid receptor 1-related disorders ASTRAZENECA AB (SE) 2009-09-02 CN disclosed