SCHEMBL28782824

SCHEMBL28782824

C(#Cc1ccccc1)CNc1ccc2ccccc2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.55
ALDH1A1 P00352 3/20 0.55
CYP3A4 P08684 3/20 0.55
CYP2C19 P33261 3/20 0.55
HSD17B10 Q99714 2/20 0.55
HIF1A Q16665 2/20 0.55
CYP2C9 P11712 2/20 0.55
CYP2D6 P10635 1/20 0.55
HPGD P15428 1/20 0.46
PIN1 Q13526 1/20 0.43
GRM5 P41594 1/20 0.42
INSR P06213 1/20 0.42
IGF1R P08069 1/20 0.42
SIGMAR1 Q99720 1/20 0.41
MRGPRX4 Q96LA9 1/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 2/20 0.40
RAB9A P51151 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28546126 0.80 GRM5 (0.54) CYP1A2ALDH1A1CYP3A4CYP2C19CYP2C9
SCHEMBL29712697 0.77 MAPT (0.53) CYP1A2ALDH1A1CYP3A4CYP2C19CYP2C9
SCHEMBL29712668 0.77 MAPT (0.55) CYP1A2ALDH1A1CYP3A4CYP2C19CYP2C9
SCHEMBL29712684 0.77 ALDH1A1 (0.54) CYP1A2ALDH1A1CYP3A4CYP2C19HSD17B10
SCHEMBL29712663 0.76 GRM5 (0.44) CYP1A2CYP3A4CYP2C19CYP2C9GRM5
SCHEMBL29712674 0.76 PYCR1 (0.50) CYP1A2ALDH1A1CYP3A4CYP2C19CYP2C9
SCHEMBL29712650 0.76 EGLN1 (0.46) CYP1A2ALDH1A1CYP3A4CYP2C19CYP2C9
SCHEMBL29543167 0.75 ALDH1A1 (0.53) CYP1A2ALDH1A1CYP3A4CYP2C19HSD17B10
SCHEMBL29712670 0.75 GRM5 (0.59) CYP1A2ALDH1A1CYP3A4CYP2C19CYP2C9
SCHEMBL7424374 0.75 ALDH1A1 (0.62) CYP1A2ALDH1A1CYP3A4CYP2C19HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110467572-B Synthetic method of 3-sulfonyl quinoline derivative 温州大学 2022-07-08 CN disclosed