SCHEMBL28784158

SCHEMBL28784158

O=Cc1cc(-c2ccccc2)nc2cccnc12

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 9/20 0.65
NPC1 O15118 2/20 0.43
DHODH Q02127 3/20 0.42
KDM4E B2RXH2 2/20 0.42
LMNA P02545 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
PDE10A Q9Y233 1/20 0.42
MEN1 O00255 1/20 0.42
HSP90AA1 P07900 1/20 0.42
IDO1 P14902 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
ACHE P22303 1/20 0.41
PDE4A P27815 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2169577 0.79 ACHE (0.56) DHODHKDM4ELMNASMN1; SMN2PDE10A
SCHEMBL18020161 0.79 TOP1 (1.00) TOP1NPC1DHODHACHE
SCHEMBL30612203 0.76 L3MBTL1 (0.45) TOP1NPC1KDM4ELMNASMN1; SMN2
SCHEMBL26106623 0.76 L3MBTL1 (0.45) TOP1NPC1KDM4ELMNASMN1; SMN2
SCHEMBL14034292 0.76 TOP1 (0.42) TOP1NPC1DHODHKDM4ELMNA
SCHEMBL26649401 0.74 DHODH (0.57) NPC1DHODHKDM4ELMNASMN1; SMN2
SCHEMBL19844332 0.72 TOP1 (0.82) TOP1DHODHKDM4ELMNAMEN1
SCHEMBL10964842 0.71 METAP1 (0.54) NPC1DHODHKDM4ELMNASMN1; SMN2
SCHEMBL27509270 0.71 TLR8 (0.40) TOP1NPC1KDM4EMEN1HSP90AA1
SCHEMBL27939580 0.70 CYP19A1 (0.56) TOP1NPC1DHODHKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101583280-B Novel hydrophilic derivatives of 2-aryl-4-quinolones as anticancer agents UNIV CHINA MEDICAL 2013-04-24 CN disclosed
CN-101583280-A Novel hydrophilic derivatives of 2-aryl-4-quinolones as anticancer agents UNIV CHINA MEDICAL (CN) 2009-11-18 CN disclosed