SCHEMBL18020161

SCHEMBL18020161

c1ccc(-c2cc(-c3ccccc3)c3ncccc3n2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 10/20 1.00
NPC1 O15118 1/20 0.49
ACHE P22303 1/20 0.47
DHODH Q02127 3/20 0.47
MAPK1 P28482 2/20 0.47
TSHR P16473 1/20 0.47
HSD17B10 Q99714 1/20 0.47
ACACA Q13085 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19844332 0.91 TOP1 (0.82) TOP1DHODHACACA
SCHEMBL19986174 0.83 TOP1 (0.71) TOP1DHODHHSD17B10
SCHEMBL19986179 0.80 TOP1 (0.67) TOP1DHODHHSD17B10
SCHEMBL18292076 0.80 TOP1 (0.64) TOP1DHODHMAPK1TSHRHSD17B10
SCHEMBL28784158 0.79 TOP1 (0.65) TOP1NPC1ACHEDHODH
SCHEMBL23946379 0.75 TOP1 (0.60) TOP1NPC1MAPK1
SCHEMBL1042853 0.75 ACACA (0.72) TOP1ACHEDHODHMAPK1ACACA
SCHEMBL29399315 0.75 ACACA (0.72) TOP1ACHEDHODHMAPK1ACACA
SCHEMBL28659827 0.75 TOP1 (0.59) TOP1NPC1MAPK1TSHR
SCHEMBL19986177 0.74 TOP1 (0.59) TOP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016128103-A1 ELECTRONIC DEVICE CONTAINING CYCLIC LACTAMS MERCK PATENT GMBH (DE) 2016-08-18 WO disclosed