SCHEMBL28784267

SCHEMBL28784267

Cc1c(C(N)=O)cccc1-c1ccccc1F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.50
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
BCAT2 O15382 1/20 0.46
KEAP1 Q14145 1/20 0.45
NFE2L2 Q16236 1/20 0.45
GRM2 Q14416 1/20 0.45
JAK2 O60674 1/20 0.44
CES2 O00748 2/20 0.42
CES1 P23141 2/20 0.42
MYC P01106 1/20 0.42
CDC7 O00311 1/20 0.42
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPT P10636 2/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PDK2 Q15119 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3837773 0.88 JAK2 (0.48) PARP1NPC1RAB9ABCAT2KEAP1
SCHEMBL30471810 0.87 BCAT2 (0.52) PARP1BCAT2KEAP1NFE2L2MYC
SCHEMBL2113823 0.83 NPC1 (0.59) PARP1NPC1RAB9ABCAT2KEAP1
SCHEMBL2468641 0.83 ESR1 (0.51) PARP1NPC1RAB9ACES2CES1
SCHEMBL3135445 0.82 MYC (0.53) PARP1BCAT2KEAP1NFE2L2MYC
Hydrochloric Acid SCHEMBL27873130 0.82 ESR1 (0.50) PARP1NPC1RAB9ACES2CES1
SCHEMBL6389895 0.81 KDM4E (0.57) PARP1NPC1RAB9ABCAT2KEAP1
SCHEMBL27725563 0.80 KEAP1 (0.58) PARP1NPC1RAB9ABCAT2KEAP1
SCHEMBL5478290 0.80 PARP1 (0.45) PARP1NPC1RAB9ABCAT2KEAP1
SCHEMBL6307908 0.79 BCAT2 (0.65) PARP1NPC1RAB9ABCAT2KEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101790313-A Compound (I) SMITHKLINE BEECHAM CORP 2010-07-28 CN disclosed